Modeling, synthesis and biological evaluation of potential retinoid X receptor-selective agonists: novel halogenated analogues of 4-[1-(3,5,5,8,8-pentamethyl-5,6,7,8-tetrahydro-2-naphthyl)ethynyl]benzoic acid (bexarotene)
潜在类视黄醇X受体选择性激动剂的建模、合成和生物学评价:4-[1-(3,5,5,8,8-五甲基-5,6,7,8-四氢-2-萘基)乙炔基]苯甲酸(贝沙罗汀)的新型卤代类似物
期刊:ChemMedChem
影响因子:3.4
doi:10.1002/cmdc.201200319
Furmick, Julie K; Kaneko, Ichiro; Walsh, Angela N; Yang, Joanna; Bhogal, Jaskaran S; Gray, Geoffrey M; Baso, Juan C; Browder, Drew O; Prentice, Jessica L S; Montano, Luis A; Huynh, Chanh C; Marcus, Lisa M; Tsosie, Dorian G; Kwon, Jungeun S; Quezada, Alexis; Reyes, Nicole M; Lemming, Brittney; Saini, Puneet; van der Vaart, Arjan; Groy, Thomas L; Marshall, Pamela A; Jurutka, Peter W; Wagner, Carl E