日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of Pyrazole-Based Positron Emission Tomography Agent that Maps Histone Deacetylase 6 (HDAC6) in the Nonhuman Primate Brain

发现一种基于吡唑的正电子发射断层扫描显像剂,可用于绘制非人灵长类动物脑内组蛋白去乙酰化酶6 (HDAC6) 的分布图

Yamasaki, Tomoteru; Ohyabu, Norio; Wakabayashi, Takeshi; Ibáñez, Ignacio; Iwanaga, Kouichi; Yamamoto, Satoshi; Hattori, Masahiko; Sugita, Taku; Terada, Michiko; Onishi, Tomohiro; Sato, Sho; Kosugi, Yohei; Takano, Akihiro; McQuade, Paul; Maru, Takamitsu; Inui, Naomi; Fujinaga, Masayuki; Mori, Wakana; Nagai, Yuji; Seki, Chie; Uchida, Shoko; Minamimoto, Takafumi; Higuchi, Makoto; Fushimi, Makoto; Zhang, Ming-Rong

Regiodivergent Nucleophilic Fluorination under Hydrogen Bonding Catalysis: A Computational and Experimental Study

氢键催化下的区域发散亲核氟化反应:计算与实验研究

Horwitz, Matthew A; Dürr, Alexander B; Afratis, Konstantinos; Chen, Zijun; Soika, Julia; Christensen, Kirsten E; Fushimi, Makoto; Paton, Robert S; Gouverneur, Véronique

Scaffold Hopping and Optimization of Small Molecule Soluble Adenyl Cyclase Inhibitors Led by Free Energy Perturbation

自由能扰动引导的小分子可溶性腺苷酸环化酶抑制剂的骨架跃迁和优化

Sun, Shan; Fushimi, Makoto; Rossetti, Thomas; Kaur, Navpreet; Ferreira, Jacob; Miller, Michael; Quast, Jonathan; van den Heuvel, Joop; Steegborn, Clemens; Levin, Lonny R; Buck, Jochen; Myers, Robert W; Kargman, Stacia; Liverton, Nigel; Meinke, Peter T; Huggins, David J

Discovery of TDI-10229: A Potent and Orally Bioavailable Inhibitor of Soluble Adenylyl Cyclase (sAC, ADCY10)

TDI-10229 的发现:一种强效且口服生物利用度高的可溶性腺苷酸环化酶 (sAC, ADCY10) 抑制剂

Fushimi, Makoto; Buck, Hannes; Balbach, Melanie; Gorovyy, Anna; Ferreira, Jacob; Rossetti, Thomas; Kaur, Navpreet; Levin, Lonny R; Buck, Jochen; Quast, Jonathan; van den Heuvel, Joop; Steegborn, Clemens; Finkin-Groner, Efrat; Kargman, Stacia; Michino, Mayako; Foley, Michael A; Miller, Michael; Liverton, Nigel J; Huggins, David J; Meinke, Peter T

Prediction of Compound Bioactivities Using Heat-Diffusion Equation.

利用热扩散方程预测化合物生物活性

Hidaka Tadashi, Imamura Keiko, Hioki Takeshi, Takagi Terufumi, Giga Yoshikazu, Giga Mi-Ho, Nishimura Yoshiteru, Kawahara Yoshinobu, Hayashi Satoru, Niki Takeshi, Fushimi Makoto, Inoue Haruhisa

Optimization of lead compounds into on-demand, nonhormonal contraceptives: leveraging a public-private drug discovery institute collaboration†

将先导化合物优化为按需服用的非激素避孕药:利用公私合作药物研发机构†

Balbach, Melanie; Fushimi, Makoto; Huggins, David J; Steegborn, Clemens; Meinke, Peter T; Levin, Lonny R; Buck, Jochen