日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Systematic pharmacological analysis of agonistic and antagonistic fibroblast growth factor receptor 1 MAbs reveals a similar unique mode of action

激动剂和拮抗剂成纤维细胞生长因子受体 1 MAb 的系统药理学分析揭示了相似的独特作用方式

Jocelyn Chan, Joyce Chan, Lily Shao, Scott S Stawicki, Victoria C Pham, Rob W Akita, Marc Hafner, Lisa Crocker, Kebing Yu, James T Koerber, Gabriele Schaefer, Laetitia Comps-Agrar

ERBB3 and IGF1R Signaling Are Required for Nrf2-Dependent Growth in KEAP1-Mutant Lung Cancer

ERBB3 和 IGF1R 信号传导是 KEAP1 突变肺癌中 Nrf2 依赖性生长所必需的

Steffan Vartanian #, James Lee #, Christiaan Klijn, Florian Gnad, Maria Bagniewska, Gabriele Schaefer, Donglu Zhang, Jenille Tan, Sara A Watson, Liling Liu, Honglin Chen, Yuxin Liang, Colin Watanabe, Trinna Cuellar, David Kan, Ryan J Hartmaier, Ted Lau, Michael R Costa, Scott E Martin, Mark Merchant

NRG1 is a critical regulator of differentiation in TP63-driven squamous cell carcinoma

NRG1是TP63驱动的鳞状细胞癌分化过程中的关键调节因子。

Ganapati V Hegde ,Cecile de la Cruz ,Jennifer M Giltnane ,Lisa Crocker ,Avinashnarayan Venkatanarayan ,Gabriele Schaefer ,Debra Dunlap ,Joerg D Hoeck ,Robert Piskol ,Florian Gnad ,Zora Modrusan ,Frederic J de Sauvage ,Christian W Siebel ,Erica L Jackson

Combined MEK and ERK inhibition overcomes therapy-mediated pathway reactivation in RAS mutant tumors

MEK 和 ERK 联合抑制可克服 RAS 突变肿瘤中治疗介导的通路再激活

Mark Merchant, John Moffat, Gabriele Schaefer, Jocelyn Chan, Xi Wang, Christine Orr, Jason Cheng, Thomas Hunsaker, Lily Shao, Stephanie J Wang, Marie-Claire Wagle, Eva Lin, Peter M Haverty, Sheerin Shahidi-Latham, Hai Ngu, Margaret Solon, Jeffrey Eastham-Anderson, Hartmut Koeppen, Shih-Min A Huang, 

High cell-surface density of HER2 deforms cell membranes

HER2 在细胞表面的高密度导致细胞膜变形

Inhee Chung, Mike Reichelt, Lily Shao, Robert W Akita, Hartmut Koeppen, Linda Rangell, Gabriele Schaefer, Ira Mellman, Mark X Sliwkowski

Advanced Parameters of Cardiac Mechanics in Children with CKD: The 4C Study

慢性肾脏病患儿心脏力学高级参数:4C 研究

Chinali, Marcello; Matteucci, Maria Chiara; Franceschini, Alessio; Doyon, Anke; Pongiglione, Giacomo; Rinelli, Gabriele; Schaefer, Franz

Dual targeting of HER2-positive cancer with trastuzumab emtansine and pertuzumab: critical role for neuregulin blockade in antitumor response to combination therapy

曲妥珠单抗 emtansine 和帕妥珠单抗双重靶向 HER2 阳性癌症:神经调节蛋白阻断在联合治疗的抗肿瘤反应中起着关键作用

Gail D Lewis Phillips, Carter T Fields, Guangmin Li, Donald Dowbenko, Gabriele Schaefer, Kathy Miller, Fabrice Andre, Howard A Burris 3rd, Kathy S Albain, Nadia Harbeck, Veronique Dieras, Diana Crivellari, Liang Fang, Ellie Guardino, Steven R Olsen, Lisa M Crocker, Mark X Sliwkowski

Noncovalent wild-type-sparing inhibitors of EGFR T790M

EGFR T790M 的非共价野生型保留抑制剂

Ho-June Lee, Gabriele Schaefer, Timothy P Heffron, Lily Shao, Xiaofen Ye, Steve Sideris, Shiva Malek, Emily Chan, Mark Merchant, Hank La, Savita Ubhayakar, Robert L Yauch, Valentina Pirazzoli, Katerina Politi, Jeff Settleman

Hepatitis C virus induces epidermal growth factor receptor activation via CD81 binding for viral internalization and entry

丙型肝炎病毒通过 CD81 结合诱导表皮生长因子受体活化,从而实现病毒内化和进入

Jingyu Diao, Homer Pantua, Hai Ngu, Laszlo Komuves, Lauri Diehl, Gabriele Schaefer, Sharookh B Kapadia

LUZ-Y, a novel platform for the mammalian cell production of full-length IgG-bispecific antibodies

LUZ-Y,一种用于哺乳动物细胞生产全长IgG双特异性抗体的新型平台

Bernd J Wranik ,Erin L Christensen, Gabriele Schaefer, Janet K Jackman, Andrew C Vendel, Dan Eaton