Omecamtiv mecarbil and Mavacamten target the same myosin pocket despite opposite effects in heart contraction
Omecamtiv mecarbil 和 Mavacamten 针对的是相同的肌球蛋白袋,尽管它们在心脏收缩中的作用相反
期刊:Nature Communications
影响因子:14.7
doi:10.1038/s41467-024-47587-9
Daniel Auguin #, Julien Robert-Paganin #, Stéphane Réty, Carlos Kikuti, Amandine David, Gabriele Theumer, Arndt W Schmidt, Hans-Joachim Knölker, Anne Houdusse