日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Antimalarial Peptide and Polyketide Natural Products from the Fijian Marine Cyanobacterium Moorea producens

斐济海洋蓝藻 Moorea 产生的抗疟肽和聚酮天然产物

Anne Marie Sweeney-Jones, Kerstin Gagaring, Jenya Antonova-Koch, Hongyi Zhou, Nazia Mojib, Katy Soapi, Jeffrey Skolnick, Case W McNamara, Julia Kubanek

Probing the Open Global Health Chemical Diversity Library for Multistage-Active Starting Points for Next-Generation Antimalarials

探索开放全球健康化学多样性库,寻找下一代抗疟药物的多阶段活性起点

Matthew Abraham, Kerstin Gagaring, Marisa L Martino, Manu Vanaerschot, David M Plouffe, Jaeson Calla, Karla P Godinez-Macias, Alan Y Du, Melanie Wree, Yevgeniya Antonova-Koch, Korina Eribez, Madeline R Luth, Sabine Ottilie, David A Fidock, Case W McNamara, Elizabeth A Winzeler

Modular, stereocontrolled C(β)-H/C(α)-C activation of alkyl carboxylic acids

烷基羧酸的模块化、立体控制的C(β)-H/C(α)-C活化

Shang, Ming; Feu, Karla S; Vantourout, Julien C; Barton, Lisa M; Osswald, Heather L; Kato, Nobutaka; Gagaring, Kerstin; McNamara, Case W; Chen, Gang; Hu, Liang; Ni, Shengyang; Fernández-Canelas, Paula; Chen, Miao; Merchant, Rohan R; Qin, Tian; Schreiber, Stuart L; Melillo, Bruno; Yu, Jin-Quan; Baran, Phil S

Antibacterial Oligomeric Polyphenols from the Green Alga Cladophora socialis

来自绿藻Cladophora socialis的抗菌低聚多酚

Lavoie, Serge; Sweeney-Jones, Anne Marie; Mojib, Nazia; Dale, Brandon; Gagaring, Kerstin; McNamara, Case W; Quave, Cassandra L; Soapi, Katy; Kubanek, Julia

Peyssonnosides A-B, Unusual Diterpene Glycosides with a Sterically Encumbered Cyclopropane Motif: Structure Elucidation Using an Integrated Spectroscopic and Computational Workflow

Peyssonnosides AB,具有空间位阻环丙烷基序的不寻常二萜糖苷:利用整合光谱和计算工作流程进行结构解析

Khatri Chhetri, Bhuwan; Lavoie, Serge; Sweeney-Jones, Anne Marie; Mojib, Nazia; Raghavan, Vijay; Gagaring, Kerstin; Dale, Brandon; McNamara, Case W; Soapi, Katy; Quave, Cassandra L; Polavarapu, Prasad L; Kubanek, Julia

Open-source discovery of chemical leads for next-generation chemoprotective antimalarials

利用开源方式发现下一代化学保护性抗疟药物的先导化合物

Antonova-Koch, Yevgeniya; Meister, Stephan; Abraham, Matthew; Luth, Madeline R; Ottilie, Sabine; Lukens, Amanda K; Sakata-Kato, Tomoyo; Vanaerschot, Manu; Owen, Edward; Jado, Juan Carlos; Maher, Steven P; Calla, Jaeson; Plouffe, David; Zhong, Yang; Chen, Kaisheng; Chaumeau, Victor; Conway, Amy J; McNamara, Case W; Ibanez, Maureen; Gagaring, Kerstin; Serrano, Fernando Neria; Eribez, Korina; Taggard, Cullin McLean; Cheung, Andrea L; Lincoln, Christie; Ambachew, Biniam; Rouillier, Melanie; Siegel, Dionicio; Nosten, François; Kyle, Dennis E; Gamo, Francisco-Javier; Zhou, Yingyao; Llinás, Manuel; Fidock, David A; Wirth, Dyann F; Burrows, Jeremy; Campo, Brice; Winzeler, Elizabeth A

High-Throughput Luciferase-Based Assay for the Discovery of Therapeutics That Prevent Malaria

基于高通量荧光素酶的检测方法用于发现预防疟疾的治疗方法

Justine Swann, Victoria Corey, Christina A Scherer, Nobutaka Kato, Eamon Comer, Micah Maetani, Yevgeniya Antonova-Koch, Christin Reimer, Kerstin Gagaring, Maureen Ibanez, David Plouffe, Anne-Marie Zeeman, Clemens H M Kocken, Case W McNamara, Stuart L Schreiber, Brice Campo, Elizabeth A Winzeler, Ste

Mutations in the P-type cation-transporter ATPase 4, PfATP4, mediate resistance to both aminopyrazole and spiroindolone antimalarials

P型阳离子转运蛋白ATPase 4 (PfATP4) 的突变介导了对氨基吡唑和螺吲哚酮类抗疟药的耐药性。

Flannery, Erika L; McNamara, Case W; Kim, Sang Wan; Kato, Tomoyo Sakata; Li, Fengwu; Teng, Christine H; Gagaring, Kerstin; Manary, Micah J; Barboa, Rachel; Meister, Stephan; Kuhen, Kelli; Vinetz, Joseph M; Chatterjee, Arnab K; Winzeler, Elizabeth A

KAI407, a potent non-8-aminoquinoline compound that kills Plasmodium cynomolgi early dormant liver stage parasites in vitro

KAI407 是一种强效的非 8-氨基喹啉类化合物,可在体外杀死猴疟原虫早期休眠肝期寄生虫。

Zeeman, Anne-Marie; van Amsterdam, Sandra M; McNamara, Case W; Voorberg-van der Wel, Annemarie; Klooster, Els J; van den Berg, Alexander; Remarque, Edmond J; Plouffe, David M; van Gemert, Geert-Jan; Luty, Adrian; Sauerwein, Robert; Gagaring, Kerstin; Borboa, Rachel; Chen, Zhong; Kuhen, Kelli; Glynne, Richard J; Chatterjee, Arnab K; Nagle, Advait; Roland, Jason; Winzeler, Elizabeth A; Leroy, Didier; Campo, Brice; Diagana, Thierry T; Yeung, Bryan K S; Thomas, Alan W; Kocken, Clemens H M

KAF156 is an antimalarial clinical candidate with potential for use in prophylaxis, treatment, and prevention of disease transmission

KAF156 是一种抗疟临床候选药物,具有用于预防、治疗和防止疾病传播的潜力。

Kelli L Kuhen, Arnab K Chatterjee, Matthias Rottmann, Kerstin Gagaring, Rachel Borboa, Jennifer Buenviaje, Zhong Chen, Carolyn Francek, Tao Wu, Advait Nagle, S Whitney Barnes, David Plouffe, Marcus C S Lee, David A Fidock, Wouter Graumans, Marga van de Vegte-Bolmer, Geert J van Gemert, Grennady Wirj