日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Development of Squaramides as Allosteric Modulators of the CB(1) Receptor: Synthesis, Computational Studies, Biological Characterization, and Effects against Cocaine-Induced Behavioral Sensitization and Reinstatement in Rats.

方酰胺作为 CB(1) 受体变构调节剂的开发:合成、计算研究、生物学表征以及对大鼠可卡因诱导的行为敏感化和复吸的影响

Nguyen Thuy, Decker Ann M, Barrus Daniel G, Song Chi Hyuck, Liu Jianfeng, Gamage Thomas F, Harris Danni L, Li Jun-Xu, Zhang Yanan

Exploring determinants of agonist efficacy at the CB1 cannabinoid receptor: Analogues of the synthetic cannabinoid receptor agonist EG-018

探索CB1大麻素受体激动剂效力的决定因素:合成大麻素受体激动剂EG-018的类似物

Finlay, David B; Nguyen, Thuy; Gamage, Thomas F; Chen, Shuli; Barrus, Daniel G; Patel, Purvi R; Thomas, Brian F; Wiley, Jenny L; Zhang, Yanan; Glass, Michelle

Sex, species and age: Effects of rodent demographics on the pharmacology of ∆(9)-tetrahydrocanabinol

性别、物种和年龄:啮齿动物种群特征对Δ(9)-四氢卡那宾醇药理学的影响

Wiley, Jenny L; Barrus, Daniel G; Farquhar, Charlotte E; Lefever, Timothy W; Gamage, Thomas F

Diarylureas Containing 5-Membered Heterocycles as CB(1) Receptor Allosteric Modulators: Design, Synthesis, and Pharmacological Evaluation

含五元杂环的二芳基脲类化合物作为CB(1)受体变构调节剂:设计、合成及药理学评价

Nguyen, Thuy; Gamage, Thomas F; Decker, Ann M; German, Nadezhda; Langston, Tiffany L; Farquhar, Charlotte E; Kenakin, Terry P; Wiley, Jenny L; Thomas, Brian F; Zhang, Yanan

Synthetic Cannabinoid Hydroxypentyl Metabolites Retain Efficacy at Human Cannabinoid Receptors

合成大麻素羟戊基代谢物在人体大麻素受体上仍保持效力

Gamage, Thomas F; Farquhar, Charlotte E; McKinnie, Ryan J; Kevin, Richard C; McGregor, Iain S; Trudell, Mark L; Wiley, Jenny L; Thomas, Brian F

Design, synthesis, and analysis of antagonists of GPR55: Piperidine-substituted 1,3,4-oxadiazol-2-ones

GPR55拮抗剂的设计、合成和分析:哌啶取代的1,3,4-恶二唑-2-酮

Meza-Aviña, Maria Elena; Lingerfelt, Mary A; Console-Bram, Linda M; Gamage, Thomas F; Sharir, Haleli; Gettys, Kristen E; Hurst, Dow P; Kotsikorou, Evangelia; Shore, Derek M; Caron, Marc G; Rao, Narasinga; Barak, Larry S; Abood, Mary E; Reggio, Patricia H; Croatt, Mitchell P

The endocannabinoid system: role in energy regulation

内源性大麻素系统:在能量调节中的作用

Gamage, Thomas F; Lichtman, Aron H