日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Library docking for Cannabinoid-2 Receptor ligands

大麻素-2受体配体的库对接

Rachman, Moira M; Iliopoulos-Tsoutsouvas, Christos; Sacco, Michael D; Xu, Xinyu; Wu, Cheng-Guo; Santos, Emma; Glenn, Isabella S; Paris, Lu; Cahill, Michelle K; Ganapathy, Suthakar; Tummino, Tia A; Moroz, Yurii S; Radchenko, Dmytro S; Okorie, Meri; Tawfik, Vivianne; Irwin, John J; Makriyannis, Alexandros; Skiniotis, Georgios; Shoichet, Brian K

Virtual library docking for cannabinoid-1 receptor agonists with reduced side effects.

针对副作用较小的 1 型大麻素受体激动剂的虚拟库对接

Tummino Tia A, Iliopoulos-Tsoutsouvas Christos, Braz Joao M, O'Brien Evan S, Stein Reed M, Craik Veronica, Tran Ngan K, Ganapathy Suthakar, Liu Fangyu, Shiimura Yuki, Tong Fei, Ho Thanh C, Radchenko Dmytro S, Moroz Yurii S, Rosado Sian Rodriguez, Bhardwaj Karnika, Benitez Jorge, Liu Yongfeng, Kandasamy Herthana, Normand Claire, Semache Meriem, Sabbagh Laurent, Glenn Isabella, Irwin John J, Kumar Kaavya Krishna, Makriyannis Alexandros, Basbaum Allan I, Shoichet Brian K

Novel Tetraolefinic Chain Phenyl Substituted Endocannabinoid Probes.

新型四烯烃链苯基取代内源性大麻素探针。

Georgiadis Markos-Orestis, Ji Lipin, Tong Fei, Dang Vuong Q, Ferreira Luana Assis, Faragher Alexandra, Tran Ngan, Sadybekov Anastasiia V, Ganapathy Suthakar, Zvonok Nikolai, Katritch Vsevolod, Hohmann Andrea G, Bohn Laura M, Makriyannis Alexandros, Nikas Spyros P

Large library docking for cannabinoid-1 receptor agonists with reduced side effects

针对副作用较小的1型大麻素受体激动剂的大型化合物库对接

Tummino, Tia A; Iliopoulos-Tsoutsouvas, Christos; Braz, Joao M; O'Brien, Evan S; Stein, Reed M; Craik, Veronica; Tran, Ngan K; Ganapathy, Suthakar; Liu, Fangyu; Shiimura, Yuki; Tong, Fei; Ho, Thanh C; Radchenko, Dmytro S; Moroz, Yurii S; Rosado, Sian Rodriguez; Bhardwaj, Karnika; Benitez, Jorge; Liu, Yongfeng; Kandasamy, Herthana; Normand, Claire; Semache, Meriem; Sabbagh, Laurent; Glenn, Isabella; Irwin, John J; Kumar, Kaavya Krishna; Makriyannis, Alexandros; Basbaum, Allan I; Shoichet, Brian K

Correction: Suppression of PKC causes oncogenic stress for triggering apoptosis in cancer cells

更正:抑制蛋白激酶C (PKC) 会导致致癌应激,从而触发癌细胞凋亡。

Ganapathy, Suthakar; Peng, Bo; Shen, Ling; Yu, Tianqi; Lafontant, Jean; Li, Ping; Xiong, Rui; Makriyannis, Alexandros; Chen, Changyan

PKC is an indispensable factor in promoting environmental toxin chromium-mediated transformation and drug resistance

蛋白激酶C (PKC) 是促进环境毒素铬介导的转化和耐药性的一个不可或缺的因素。

Ganapathy, Suthakar; Liu, Jian; Yu, Tianqi; Xiong, Rui; Zhang, Qiang; Makriyannis, Alexandros; Chen, Changyan

A lethal synergy induced by phellinus linteus and camptothecin11 in colon cancer cells

裂叶木虱和喜树碱11在结肠癌细胞中诱导的致命协同作用

Yu, Tianqi; Ganapathy, Suthakar; Shen, Ling; Peng, Bo; Kim, Sung-Hoon; Makriyannis, Alexandros; Chen, Changyan

Suppression of PKC causes oncogenic stress for triggering apoptosis in cancer cells

抑制蛋白激酶C (PKC) 可导致致癌应激,从而触发癌细胞凋亡。

Ganapathy, Suthakar; Peng, Bo; Shen, Ling; Yu, Tianqi; Lafontant, Jean; Li, Ping; Xiong, Rui; Makriyannis, Alexandros; Chen, Changyan

Bone Morphogenetic Protein-2 (BMP-2) Activates NFATc1 Transcription Factor via an Autoregulatory Loop Involving Smad/Akt/Ca2+ Signaling

骨形态发生蛋白-2 (BMP-2) 通过涉及 Smad/Akt/Ca2+ 信号的自调节环激活 NFATc1 转录因子

Mandal, Chandi C; Das, Falguni; Ganapathy, Suthakar; Harris, Stephen E; Choudhury, Goutam Ghosh; Ghosh-Choudhury, Nandini

Ral A, via activating the mitotic checkpoint, sensitizes cells lacking a functional Nf1 to apoptosis in the absence of protein kinase C

Ral A 通过激活有丝分裂检查点,使缺乏功能性 Nf1 的细胞在缺乏蛋白激酶 C 的情况下对凋亡更加敏感。

Ganapathy, Suthakar; Fagman, Johan B; Shen, Ling; Yu, Tianqi; Zhou, Xiaodong; Dai, Wei; Makriyannis, Alexandros; Chen, Changyan