日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery, Characterization, and Optimization of a Novel Positive Allosteric Modulator-Antagonist of the D(3) Dopamine Receptor.

发现、表征和优化一种新型的D(3)多巴胺受体正向变构调节剂-拮抗剂

Moritz Amy E, Wang Feijun, Madaras Nora S, Kelley Amber M, Snyder Kirsten K, Gandhi Disha, Inbody Laura R, Akano Emmanuel O, Shi Lei, Lane J Robert, Free R Benjamin, Frankowski Kevin J, Sibley David R

Synthesis and initial pharmacology of dual-targeting ligands for putative complexes of integrin αVβ3 and PAR2

合成并初步研究了针对整合素αVβ3和PAR2假定复合物的双靶向配体

Majewski, Mark W; Gandhi, Disha M; Holyst, Trudy; Wang, Zhengli; Hernandez, Irene; Rosas, Ricardo Jr; Zhu, Jieqing; Weiler, Hartmut; Dockendorff, Chris

NMR Structural Analysis of Isolated Shaker Voltage-Sensing Domain in LPPG Micelles

LPPG胶束中分离的Shaker电压传感域的NMR结构分析

Chen, Hongbo; Pan, Junkun; Gandhi, Disha M; Dockendorff, Chris; Cui, Qiang; Chanda, Baron; Henzler-Wildman, Katherine A

The parmodulin NRD-21 is an allosteric inhibitor of PAR1 Gq signaling with improved anti-inflammatory activity and stability

帕莫德林NRD-21是一种PAR1 Gq信号通路的变构抑制剂,具有增强的抗炎活性和稳定性。

Gandhi, Disha M; Rosas, Ricardo Jr; Greve, Eric; Kentala, Kaitlin; D-R Diby, N'Guessan; Snyder, Vladyslava A; Stephans, Allison; Yeung, Teresa H W; Subramaniam, Saravanan; DiMilo, Elliot; Kurtenbach, Khia E; Arnold, Leggy A; Weiler, Hartmut; Dockendorff, Chris