3-(2,4-dichlorophenyl)-4-(1-methyl-1H-indol-3-yl)-1H-pyrrole-2,5-dione (SB216763), a glycogen synthase kinase-3 inhibitor, displays therapeutic properties in a mouse model of pulmonary inflammation and fibrosis
3-(2,4-二氯苯基)-4-(1-甲基-1H-吲哚-3-基)-1H-吡咯-2,5-二酮 (SB216763) 是一种糖原合酶激酶-3 抑制剂,在小鼠肺部炎症和纤维化模型中表现出治疗作用
期刊:Journal of Pharmacology and Experimental Therapeutics
影响因子:3.1
doi:10.1124/jpet.109.153049
Carmela Gurrieri, Francesco Piazza, Marianna Gnoato, Barbara Montini, Lucia Biasutto, Cristina Gattazzo, Enrico Brunetta, Anna Cabrelle, Francesco Cinetto, Raffaele Niero, Monica Facco, Spiridione Garbisa, Fiorella Calabrese, Gianpietro Semenzato, Carlo Agostini