Conformational Restriction of Designer Drugs Reveals Subtype-Selective and Biased CB(2) Agonists with Neuroprotective Effects.
构象限制设计药物揭示了具有神经保护作用的亚型选择性和偏向性 CB(2) 激动剂
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.5c00604
Gioé-Gallo Claudia, Ortigueira Sandra, Prieto-DÃaz Rubén, Contino Marialessandra, Azuaje Jhonny, Perrone Maria Grazia, Riganti Chiara, Alberga Domenico, Mangiatordi Giuseppe Felice, Andújar-Arias Antonio, GarcÃa-Rey Aitor, Graziano Giovanni, Stefanachi Angela, Val Cristina, MartÃnez Antón Leandro, Rebassa Joan Biel, Reza David, Selas Asier, Francavilla Fabio, Paleo M Rita, GarcÃa-Mera Xerardo, Loza M Isabel, Navarro Gemma, Brea José, Sotelo Eddy
