Discovery of lirafugratinib (RLY-4008), a highly selective irreversible small-molecule inhibitor of FGFR2
发现利拉夫格拉替尼 (RLY-4008)，一种高选择性的不可逆小分子 FGFR2 抑制剂
期刊:Proceedings of the National Academy of Sciences of the United States of America
影响因子:9.1
doi:10.1073/pnas.2317756121
Schönherr, Heike; Ayaz, Pelin; Taylor, Alexander M; Casaletto, Jessica B; Touré, B Barry; Moustakas, Demetri T; Hudson, Brandi M; Valverde, Roberto; Zhao, Songping; O'Hearn, Patrick J; Foster, Lindsey; Sharon, Dina A; Garfinkle, Sam; Giordanetto, Fabrizio; Lescarbeau, André; Kurukulasuriya, Ravi; Gerami-Moayed, Nastaran; Maglic, Dejan; Bruderek, Kamil; Naik, Gaauri; Gunaydin, Hakan; Mader, Mary M; Boezio, Alessandro A; McLean, Thomas H; Chen, Rongfeng; Wang, Yanxia; Shaw, David E; Watters, James; Bergstrom, Donald A
