日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Pyrimidone inhibitors targeting Chikungunya Virus nsP3 macrodomain by fragment-based drug design

通过基于片段的药物设计靶向基孔肯雅病毒 nsP3 大结构域的嘧啶酮抑制剂

Sixue Zhang, Atefeh Garzan, Nicole Haese, Robert Bostwick, Yohanka Martinez-Gzegozewska, Lynn Rasmussen, Daniel N Streblow, Mark T Haise, Ashish K Pathak, Corinne E Augelli-Szafran, Mousheng Wu

Interfering With DNA Decondensation as a Strategy Against Mycobacteria

干扰DNA解凝缩作为对抗分枝杆菌的策略

Scutigliani, Enzo M; Scholl, Edwin R; Grootemaat, Anita E; Khanal, Sadhana; Kochan, Jakub A; Krawczyk, Przemek M; Reits, Eric A; Garzan, Atefeh; Ngo, Huy X; Green, Keith D; Garneau-Tsodikova, Sylvie; Ruijter, Jan M; van Veen, Henk A; van der Wel, Nicole N

Optimization of pyrazole-containing 1,2,4-triazolo-[3,4-b]thiadiazines, a new class of STAT3 pathway inhibitors

吡唑类化合物1,2,4-三唑并[3,4-b]噻二嗪的优化,一类新型STAT3通路抑制剂

LaPorte, Matthew G; Wang, Zhuzhu; Colombo, Raffaele; Garzan, Atefeh; Peshkov, Vsevolod A; Liang, Mary; Johnston, Paul A; Schurdak, Mark E; Sen, Malabika; Camarco, Daniel P; Hua, Yun; Pollock, Netanya I; Lazo, John S; Grandis, Jennifer R; Wipf, Peter; Huryn, Donna M