日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Monovalent pseudo-natural products supercharge degradation of IDO1 by its native E3 KLHDC3.

单价伪天然产物可加速 IDO1 的天然 E3 KLHDC3 的降解。

Hennes Elisabeth, Lucas Belén, Scholes Natalie S, Cheng Xiu-Fen, Scott Daniel C, Bischoff Matthias, Reich Katharina, Gasper Raphael, Lucas María, Xu Teng Teng, Rossini Sofia, Pulvermacher Lisa-Marie, Dötsch Lara, Imrichova Hana, Brause Alexandra, Führer Siska, Naredla Kesava Reddy, Sievers Sonja, Kumar Kamal, Janning Petra, Orabona Ciriana, Gersch Malte, Murray Peter J, Schulman Brenda A, Winter Georg E, Ziegler Slava, Waldmann Herbert

Design, Synthesis, and Structural Evolution of Pseudo-Natural Product IDO1 Inhibitors and Degraders

拟天然产物IDO1抑制剂和降解剂的设计、合成和结构演变

Cheng, Xiu-Fen; Lucas, Belén; Lampe, Philipp; Ugel, Stefano; Chen, Suyuan; Unger, Anke; Bischoff, Matthias; Adariani, Soheila Rezaei; Naredla, Kesava Reddy; Kumar, Kamal; Schmidt, Annika; Strohmann, Carsten; Janning, Petra; Gasper, Raphael; Lucas, María; Gersch, Malte; Sievers, Sonja; Bronte, Vincenzo; Ziegler, Slava; Waldmann, Herbert

Crowdsourced biodiversity monitoring fills gaps in global plant trait mapping

众包生物多样性监测填补了全球植物性状图谱绘制的空白。

Lusk, Daniel; Wolf, Sophie; Svidzinska, Daria; Dormann, Carsten F; Kattge, Jens; Bruelheide, Helge; Sabatini, Francesco Maria; Damasceno, Gabriella; Moreno Martínez, Álvaro; Violle, Cyrille; Hending, Daniel; Hähn, Georg J A; Tabeni, Solana; Phartyal, Shyam; Gonçalves, Fernando; Kreft, Holger; Schmidt, Marco; Chen, Han; Güler, Behlül; Dolezal, Jiri; Pielech, Remigiusz; Guido, Anaclara; Dwyer, Ciara; Napoleone, Francesca; Willie, Jacob; Gasper, André Luís; Macía, Manuel J; Chytry, Milan; Lenoir, Jonathan; Thakur, Dinesh; Dengler, Jürgen; Świerszcz, Sebastian; Altman, Jan; Mucina, Ladislav; Nerlekar, Ashish N; Kakinuma, Kaoru; Rawat, Pravin; Stančić, Zvjezdana; Testolin, Riccardo; Hatim, Mohamed Z; Rodrigues, Flávio; Homeier, Jürgen; Marques, Marcia C M; McCarthy, James K; El-Sheikh, M A; Korznikov, Kirill; Gerberding, Kilian; Kattenborn, Teja

Covalent modification of a glutamic acid inspired by HaloTag technology.

受 HaloTag 技术启发,对谷氨酸进行共价修饰。

Zhang Ruirui, Liu Jie, Gasper Raphael, Unger Anke, Kaschani Farnusch, Kaiser Markus, Janning Petra, Waldmann Herbert

Targeting a Glutamic Acid in PDEδ with Fluoromethyl-Aryl Electrophiles Impairs K-Ras Signaling

用氟甲基-芳基亲电试剂靶向PDEδ中的谷氨酸会损害K-Ras信号传导

Zhang, Ruirui; Huetzen, Maxim A; Binici, Aylin; Martín-Gago, Pablo; Gasper, Raphael; Rudashevskaya, Elena; Liu, Jie; Nagaraju, Chinta; Reckzeh, Elena S; Stuedle, Alana S T; Hopff, Ann-Sophie; Mesaros, Andrea; Unger, Anke; Thelen, Melanie; Janning, Petra; Reinhardt, H Christian; Ziegler, Slava; Jachimowicz, Ron D; Waldmann, Herbert

Surface markers on supermeres outperform extracellular vesicles in colorectal cancer diagnosis

在结直肠癌诊断中,超分子表面标志物优于细胞外囊泡。

Kumar, Sonu; Sinclair, John Alex; Shi, Tiger; Kim, Gaeun; Zhu, Runyao; Gasper, Grace; Wang, Yichun; Higginbotham, James N; Zhang, Qin; Jeppesen, Dennis K; Tutanov, Oleg; Hamilton, Maxwell; Franklin, Jeffrey L; Charest, Al; Coffey, Robert J; Senapati, Satyajyoti; Chang, Hsueh-Chia

Safety and optimal timing of staged nipple-sparing mastectomy following nipple repositioning in ptotic breasts: a systematic review protocol

乳头下垂乳房乳头复位后分期保留乳头乳房切除术的安全性和最佳时机:系统评价方案

Tanas, Yousef; Gasper, Grace; Swed, Sarya; Spiegel, Aldona J

Contemporary outcomes of lower extremity vein bypass for chronic limb-threatening ischemia based on a post hoc comparison of the BEST-CLI and PREVENT III multicenter prospective randomized controlled trials

基于对 BEST-CLI 和 PREVENT III 多中心前瞻性随机对照试验的事后比较,探讨下肢静脉旁路术治疗慢性肢体缺血的最新疗效

Hussain, Mohamad A; Khan, Ali A; Menard, Matthew T; Conte, Michael S; Vouyouka, Ageliki G; Doros, Gheorghe; Strong, Michael B; Kalish, Jeffrey A; Chew, David; Gasper, Warren J; Tan, Tze-Woei; Darling, R Clement 3rd; LaMuraglia, Glenn; Rosenfield, Kenneth; Farber, Alik; Schanzer, Andres

Assessing nonresponse bias in a 30-year study of gulf war and gulf era veterans

评估一项针对海湾战争和海湾时期老兵的30年研究中的无应答偏差

Gasper, Joseph; Van de Kerckhove, Wendy; Spark, Talia; McCall, James; Mihovich, Carly; Hammer, Heather; Schneiderman, Aaron; Madden, Michele; Dursa, Erin K

Lessons from the field: implementing pharmacy services in the Tanzanian hospital setting

来自实地的经验教训:在坦桑尼亚医院环境中实施药学服务

Lambert, Maarten; Mmassy, John; Kabissi, Sungwa; Benizeth, Cecilia; Baltazary, Gasper; Maganda, Betty Allen; Taxis, Katja