Discovery of Highly Potent and Selective IRAK1 Degraders to Probe Scaffolding Functions of IRAK1 in ABC DLBCL
发现高效且选择性的 IRAK1 降解剂,用于探究 ABC DLBCL 中 IRAK1 的支架功能
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.1c00103
Liqiang Fu, Jing Zhang, Bin Shen, Linglong Kong, Yingtao Liu, Wangyang Tu, Wenqian Wang, Xin Cai, Xiaotao Wang, Na Cheng, Mingxuan Xia, Tianyuan Zhou, Qian Liu, Yanping Xu, Jennifer Yang, Paul Gavine, Ulrike Philippar, Ricardo Attar, James P Edwards, Jennifer D Venable, Xuedong Dai