Allosteric targeting of RIPK1: discovery of novel inhibitors via parallel virtual screening and structure-guided optimization
RIPK1的变构靶向:通过并行虚拟筛选和结构导向优化发现新型抑制剂
期刊:RSC Medicinal Chemistry
影响因子:3.6
doi:10.1039/d5md00317b
Vijayan, R S K; Hamilton, Matthew M; Pfaffinger, Dana E; Alvarez, Fernando G; Reyna, Naphtali J; Bardenhagen, Jennifer P; Shepard, Hannah; Rodriguez, Christian; Goodwani, Sunil; Lightfoot, Yaima; Maskos, Klaus; Johannsson, Sven; Kempf, Georg; Xu, Quanyun Alan; Neumann, Lars; Jiang, Yongying; Do, Mary Geck; Jones, Philip; Lewis, Richard T; Ray, William J; Cross, Jason B