日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Ex vivo mass spectrometry-based biodistribution analysis of an antibody-Resiquimod conjugate bearing a protease-cleavable and acid-labile linker

利用体外质谱法对带有蛋白酶可切割和酸不稳定连接子的抗体-瑞喹莫德偶联物进行生物分布分析

Bisbal Lopez, Lydia; Ravazza, Domenico; Bocci, Matilde; Zana, Aureliano; Principi, Lucrezia; Dakhel Plaza, Sheila; Galbiati, Andrea; Gilardoni, Ettore; Scheuermann, Jörg; Neri, Dario; Pignataro, Luca; Gennari, Cesare; Cazzamalli, Samuele; Dal Corso, Alberto

Visible Light-Promoted β-Functionalization of Carbonyl Compounds in the Presence of Organic Dyes

可见光促进有机染料存在下羰基化合物的β-官能化

Dolcini, Luigi; Gandini, Tommaso; Castiglioni, Riccardo; Bossi, Alberto; Penconi, Marta; Dal Corso, Alberto; Gennari, Cesare; Pignataro, Luca

Advanced Pyrrolidine-Carbamate Self-Immolative Spacer with Tertiary Amine Handle Induces Superfast Cyclative Drug Release

具有叔胺基团的先进吡咯烷-氨基甲酸酯自毁间隔基可诱导超快速循环药物释放

Dal Corso, Alberto; Frigoli, Margaux; Prevosti, Martina; Mason, Mattia; Bucci, Raffaella; Belvisi, Laura; Pignataro, Luca; Gennari, Cesare

Rational Design of Antiangiogenic Helical Oligopeptides Targeting the Vascular Endothelial Growth Factor Receptors

靶向血管内皮生长因子受体的抗血管生成螺旋寡肽的合理设计

Zanella, Simone; Bocchinfuso, Gianfranco; De Zotti, Marta; Arosio, Daniela; Marino, Franca; Raniolo, Stefano; Pignataro, Luca; Sacco, Giovanni; Palleschi, Antonio; Siano, Alvaro S; Piarulli, Umberto; Belvisi, Laura; Formaggio, Fernando; Gennari, Cesare; Stella, Lorenzo

Neutrophil Elastase Promotes Linker Cleavage and Paclitaxel Release from an Integrin-Targeted Conjugate

中性粒细胞弹性蛋白酶促进连接子裂解和紫杉醇从整合素靶向缀合物中释放

Raposo Moreira Dias, André; Pina, Arianna; Dean, Amelia; Lerchen, Hans-Georg; Caruso, Michele; Gasparri, Fabio; Fraietta, Ivan; Troiani, Sonia; Arosio, Daniela; Belvisi, Laura; Pignataro, Luca; Dal Corso, Alberto; Gennari, Cesare

Synthesis and Biological Evaluation of RGD and isoDGR-Monomethyl Auristatin Conjugates Targeting Integrin α(V) β(3)

靶向整合素α(V)β(3)的RGD和isoDGR-单甲基奥瑞他汀缀合物的合成和生物学评价

Raposo Moreira Dias, André; Bodero, Lizeth; Martins, Ana; Arosio, Daniela; Gazzola, Silvia; Belvisi, Laura; Pignataro, Luca; Steinkühler, Christian; Dal Corso, Alberto; Gennari, Cesare; Piarulli, Umberto

Conjugates of Cryptophycin and RGD or isoDGR Peptidomimetics for Targeted Drug Delivery

隐藻素与RGD或isoDGR肽模拟物的偶联物用于靶向药物递送

Borbély, Adina; Figueras, Eduard; Martins, Ana; Bodero, Lizeth; Raposo Moreira Dias, André; López Rivas, Paula; Pina, Arianna; Arosio, Daniela; Gallinari, Paola; Frese, Marcel; Steinkühler, Christian; Gennari, Cesare; Piarulli, Umberto; Sewald, Norbert

Synthesis and biological evaluation of RGD and isoDGR peptidomimetic-α-amanitin conjugates for tumor-targeting

RGD和isoDGR肽模拟物-α-鹅膏蕈碱缀合物的合成及生物学评价及其在肿瘤靶向治疗中的应用

Bodero, Lizeth; López Rivas, Paula; Korsak, Barbara; Hechler, Torsten; Pahl, Andreas; Müller, Christoph; Arosio, Daniela; Pignataro, Luca; Gennari, Cesare; Piarulli, Umberto

Insights into the Binding of Cyclic RGD Peptidomimetics to α(5)β(1) Integrin by using Live-Cell NMR And Computational Studies.

利用活细胞核磁共振和计算研究深入了解环状RGD肽模拟物与α(5)β(1)整合素的结合

Guzzetti Ileana, Civera Monica, Vasile Francesca, Arosio Daniela, Tringali Cristina, Piarulli Umberto, Gennari Cesare, Pignataro Luca, Belvisi Laura, Potenza Donatella

Synthesis, Characterization, and Biological Evaluation of a Dual-Action Ligand Targeting αvβ3 Integrin and VEGF Receptors.

靶向αvβ3整合素和VEGF受体的双作用配体的合成、表征和生物学评价

Zanella Simone, Mingozzi Michele, Dal Corso Alberto, Fanelli Roberto, Arosio Daniela, Cosentino Marco, Schembri Laura, Marino Franca, De Zotti Marta, Formaggio Fernando, Pignataro Luca, Belvisi Laura, Piarulli Umberto, Gennari Cesare