日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

From Prompt to Drug: Toward Pharmaceutical Superintelligence

从提示到药物:迈向药物超级智能

Zhavoronkov, Alex; Gennert, David; Shi, Jiye

From Prompt to Drug: Toward Pharmaceutical Superintelligence

从提示到药物:迈向药物超级智能

Tabana, Yasser; Okoye, Isobel S; Siraki, Arno; Elahi, Shokrollah; Barakat, Khaled H; Zhavoronkov, Alex; Gennert, David; Shi, Jiye

A generative AI-discovered TNIK inhibitor for idiopathic pulmonary fibrosis: a randomized phase 2a trial

一种由人工智能发现的用于治疗特发性肺纤维化的TNIK抑制剂:一项随机2a期试验

Xu, Zuojun; Ren, Feng; Wang, Ping; Cao, Jie; Tan, Chunting; Ma, Dedong; Zhao, Li; Dai, Jinghong; Ding, Yipeng; Fang, Haohui; Li, Huiping; Liu, Hong; Luo, Fengming; Meng, Ying; Pan, Pinhua; Xiang, Pingchao; Xiao, Zuke; Rao, Sujata; Satler, Carol; Liu, Sang; Lv, Yuan; Zhao, Heng; Chen, Shan; Cui, Hui; Korzinkin, Mikhail; Gennert, David; Zhavoronkov, Alex

Discovery of a bifunctional PKMYT1-targeting PROTAC empowered by AI-generation.

利用人工智能生成技术发现双功能PKMYT1靶向PROTAC。

Wang Yazhou, Wang Xiaomin, Liu Tingting, Wang Chao, Meng Qingshuo, Meng Fanye, Yu Jiaojiao, Liu Jinxin, Fan Yaya, Gennert David, Pun Frank W, Aliper Alex, Ren Feng, Zhang Man, Cai Xin, Ding Xiao, Zhavoronkov Alex

Oral ENPP1 inhibitor designed using generative AI as next generation STING modulator for solid tumors.

利用人工智能生成技术设计的口服 ENPP1 抑制剂,作为下一代 STING 调节剂用于治疗实体瘤

Pu Congying, Cui Hui, Yu Huaxing, Cheng Xin, Zhang Man, Qin Luoheng, Ning Zhilin, Zhang Wen, Chen Shan, Qian Yuhang, Wang Feng, Wang Ling, Lin Xiaoxia, Gennert David, Pun Frank W, Ren Feng, Zhavoronkov Alex