日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Unified Software Solution for Efficient SPR Data Analysis in Drug Research

药物研究中高效 SPR 数据分析的统一软件解决方案

Göran Dahl, Stephan Steigele, Per Hillertz, Anna Tigerström, Anders Egnéus, Alexander Mehrle, Martin Ginkel, Fredrik Edfeldt, Geoff Holdgate, Nichole O'Connell, Bernd Kappler, Annette Brodte, Philip B Rawlins, Gareth Davies, Eva-Lotta Westberg, Rutger H A Folmer, Stephan Heyse

Potent and selective bivalent inhibitors of BET bromodomains

强效且选择性的 BET 溴结构域双价抑制剂

Michael J Waring, Huawei Chen, Alfred A Rabow, Graeme Walker, Romel Bobby, Scott Boiko, Rob H Bradbury, Rowena Callis, Edwin Clark, Ian Dale, Danette L Daniels, Austin Dulak, Liz Flavell, Geoff Holdgate, Thomas A Jowitt, Alexey Kikhney, Mark McAlister, Jacqui Méndez, Derek Ogg, Joe Patel, Philip Pet

Structures of the human poly (ADP-ribose) glycohydrolase catalytic domain confirm catalytic mechanism and explain inhibition by ADP-HPD derivatives

人类聚(ADP-核糖)糖水解酶催化结构域的结构证实了催化机制并解释了 ADP-HPD 衍生物的抑制作用

Julie A Tucker, Neil Bennett, Claire Brassington, Stephen T Durant, Giles Hassall, Geoff Holdgate, Mark McAlister, J Willem M Nissink, Caroline Truman, Martin Watson