日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Complex I inhibitor of oxidative phosphorylation in advanced solid tumors and acute myeloid leukemia: phase I trials.

氧化磷酸化复合物 I 抑制剂在晚期实体瘤和急性髓系白血病中的应用:I 期试验

Yap Timothy A, Daver Naval, Mahendra Mikhila, Zhang Jixiang, Kamiya-Matsuoka Carlos, Meric-Bernstam Funda, Kantarjian Hagop M, Ravandi Farhad, Collins Meghan E, Francesco Maria Emilia Di, Dumbrava Ecaterina E, Fu Siqing, Gao Sisi, Gay Jason P, Gera Sonal, Han Jing, Hong David S, Jabbour Elias J, Ju Zhenlin, Karp Daniel D, Lodi Alessia, Molina Jennifer R, Baran Natalia, Naing Aung, Ohanian Maro, Pant Shubham, Pemmaraju Naveen, Bose Prithviraj, Piha-Paul Sarina A, Rodon Jordi, Salguero Carolina, Sasaki Koji, Singh Anand K, Subbiah Vivek, Tsimberidou Apostolia M, Xu Quanyun A, Yilmaz Musa, Zhang Qi, Li Yuan, Bristow Christopher A, Bhattacharjee Meenakshi B, Tiziani Stefano, Heffernan Timothy P, Vellano Christopher P, Jones Philip, Heijnen Cobi J, Kavelaars Annemieke, Marszalek Joseph R, Konopleva Marina

Allosteric SHP2 Inhibitor, IACS-13909, Overcomes EGFR-Dependent and EGFR-Independent Resistance Mechanisms toward Osimertinib

变构SHP2抑制剂IACS-13909可克服EGFR依赖性和EGFR非依赖性奥希替尼耐药机制

Sun, Yuting; Meyers, Brooke A; Czako, Barbara; Leonard, Paul; Mseeh, Faika; Harris, Angela L; Wu, Qi; Johnson, Sarah; Parker, Connor A; Cross, Jason B; Di Francesco, Maria Emilia; Bivona, Benjamin J; Bristow, Christopher A; Burke, Jason P; Carrillo, Caroline C; Carroll, Christopher L; Chang, Qing; Feng, Ningping; Gao, Guang; Gera, Sonal; Giuliani, Virginia; Huang, Justin K; Jiang, Yongying; Kang, Zhijun; Kovacs, Jeffrey J; Liu, Chiu-Yi; Lopez, Anastasia M; Ma, Xiaoyan; Mandal, Pijus K; McAfoos, Timothy; Miller, Meredith A; Mullinax, Robert A; Peoples, Michael; Ramamoorthy, Vandhana; Seth, Sahil; Spencer, Nakia D; Suzuki, Erika; Williams, Christopher C; Yu, Simon S; Zuniga, Andy M; Draetta, Giulio F; Marszalek, Joseph R; Heffernan, Timothy P; Kohl, Nancy E; Jones, Philip