日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

ARN25068, a versatile starting point towards triple GSK-3β/FYN/DYRK1A inhibitors to tackle tau-related neurological disorders

ARN25068 是三重 GSK-3β/FYN/DYRK1A 抑制剂的多功能起点,用于治疗与 tau 相关的神经系统疾病

Stefania Demuro, Conall Sauvey, Shailesh K Tripathi, Rita M C Di Martino, Da Shi, Jose A Ortega, Debora Russo, Beatrice Balboni, Barbara Giabbai, Paola Storici, Stefania Girotto, Ruben Abagyan, Andrea Cavalli

Identification of Novel GSK-3β Hits Using Competitive Biophysical Assays.

利用竞争性生物物理测定法鉴定新型 GSK-3β 先导化合物

Balboni Beatrice, Tripathi Shailesh Kumar, Veronesi Marina, Russo Debora, Penna Ilaria, Giabbai Barbara, Bandiera Tiziano, Storici Paola, Girotto Stefania, Cavalli Andrea

Known Drugs Identified by Structure-Based Virtual Screening Are Able to Bind Sigma-1 Receptor and Increase Growth of Huntington Disease Patient-Derived Cells.

通过基于结构的虚拟筛选鉴定出的已知药物能够与 Sigma-1 受体结合,并促进亨廷顿病患者来源细胞的生长

Battista Theo, Pascarella Gianmarco, Staid David Sasah, Colotti Gianni, Rosati Jessica, Fiorillo Annarita, Casamassa Alessia, Vescovi Angelo Luigi, Giabbai Barbara, Semrau Marta Stefania, Fanelli Sergio, Storici Paola, Squitieri Ferdinando, Morea Veronica, Ilari Andrea

Structural and Biochemical Analysis of the Dual Inhibition of MG-132 against SARS-CoV-2 Main Protease (Mpro/3CLpro) and Human Cathepsin-L

MG-132 对 SARS-CoV-2 主蛋白酶 (Mpro/3CLpro) 和人组织蛋白酶-L 双重抑制的结构和生化分析

Elisa Costanzi, Maria Kuzikov, Francesca Esposito, Simone Albani, Nicola Demitri, Barbara Giabbai, Marianna Camasta, Enzo Tramontano, Giulia Rossetti, Andrea Zaliani, Paola Storici

Combination of SAXS and Protein Painting Discloses the Three-Dimensional Organization of the Bacterial Cysteine Synthase Complex, a Potential Target for Enhancers of Antibiotic Action

小角X射线散射(SAXS)与蛋白质染色技术相结合,揭示了细菌半胱氨酸合成酶复合物的三维结构,该复合物是增强抗生素作用的潜在靶点。

Rosa, Brenda; Marchetti, Marialaura; Paredi, Gianluca; Amenitsch, Heinz; Franko, Nina; Benoni, Roberto; Giabbai, Barbara; De Marino, Maria Giovanna; Mozzarelli, Andrea; Ronda, Luca; Storici, Paola; Campanini, Barbara; Bettati, Stefano

A covalent PIN1 inhibitor selectively targets cancer cells by a dual mechanism of action

共价 PIN1 抑制剂通过双重作用机制选择性地靶向癌细胞

Elena Campaner, Alessandra Rustighi, Alessandro Zannini, Alberto Cristiani, Silvano Piazza, Yari Ciani, Ori Kalid, Gali Golan, Erkan Baloglu, Sharon Shacham, Barbara Valsasina, Ulisse Cucchi, Agnese Chiara Pippione, Marco Lucio Lolli, Barbara Giabbai, Paola Storici, Paolo Carloni, Giulia Rossetti, F

Generation of functional HLA-DR*1101 tetramers receptive for loading with pathogen- or tumour-derived synthetic peptides

生成可加载病原体或肿瘤来源合成肽的功能性HLA-DR*1101四聚体

Moro, Monica; Cecconi, Virginia; Martinoli, Chiara; Dallegno, Eliana; Giabbai, Barbara; Degano, Massimo; Glaichenhaus, Nicholas; Protti, Maria Pia; Dellabona, Paolo; Casorati, Giulia