日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Optimization and Characterization of N-Acetamide Indoles as Antimalarials That Target PfATP4

优化和表征靶向 PfATP4 的 N-乙酰胺吲哚类抗疟药

Awalt, Jon Kyle; Ooi, Zi Kang; Ashton, Trent D; Mansouri, Mahta; Calic, Petar P S; Zhou, Qingmiao; Vasanthan, Santhya; Lee, Serena; Loi, Katie; Jarman, Kate E; Penington, Jocelyn S; Qiu, Deyun; Zhang, Xinxin; Lehane, Adele M; Mao, Emma Y; Gancheva, Maria R; Wilson, Danny W; Giannangelo, Carlo; MacRaild, Christopher A; Creek, Darren J; Yeo, Tomas; Sheth, Tanaya; Fidock, David A; Churchyard, Alisje; Baum, Jake; Famodimu, Mufuliat T; Delves, Michael J; Kristan, Mojca; Stewart, Lindsay; Sutherland, Colin J; Coyle, Rachael; Jagoe, Hannah; Lee, Marcus C S; Chowdury, Mrittika; de Koning-Ward, Tania F; Baud, Delphine; Brand, Stephen; Jackson, Paul F; Cowman, Alan F; Dans, Madeline G; Sleebs, Brad E

Testing the applicability of a governance checklist for high-risk AI-based learning outcome assessment in Italian universities under the EU AI act annex III

根据欧盟人工智能法案附件三,测试治理清单在意大利大学高风险人工智能学习成果评估中的适用性

Manganello, Flavio; Nico, Alberto; Ragusa, Martina; Boccuzzi, Giannangelo

Characterizing the quick-killing mechanism of action of azithromycin analogs against malaria parasites

阐明阿奇霉素类似物对疟原虫的快速杀灭机制

Mao, Emma Y; Nguyen, William; Jana, Gouranga P; Maity, Bikash C; Pazicky, Samuel; Giannangelo, Carlo; Reader, Janette; Famodimu, Mufuliat T; Birkholtz, Lyn-Marie; Delves, Michael J; Creek, Darren J; Bozdech, Zbynek; Laleu, Benoît; Burrows, Jeremy N; Sleebs, Brad E; Gancheva, Maria R; Wilson, Danny W

Novel heterospirocyclic antimalarials with activity against artemisinin- and multidrug-resistant P. falciparum malaria

新型杂螺环抗疟药对青蒿素耐药和多重耐药的恶性疟原虫疟疾具有活性

Theodoridis, Liana; Giannangelo, Carlo; El-Saafin, Farrah; Prabhath, Mr Ranga; Macraild, Christopher A; Sharma, Pallavi; Merino, Delphine; Creek, Darren J; Carvalho, Teresa G

Validation of solvent proteome profiling for antimalarial drug target deconvolution

溶剂蛋白质组分析在抗疟药物靶点解卷积中的验证

Ji, Yijia; Morrow, Joshua P; MacRaild, Christopher A; Zhang, Haijian; Giannangelo, Carlo; Schittenhelm, Ralf B; Creek, Darren J; Siddiqui, Ghizal

A Transformative Innovation to Clinical Coding for Better Data and Less Burden

临床编码的变革性创新,带来更优质的数据和更轻的负担

Pine, Michael; Giannangelo, Kathy; Hobson, Charles; Tompkins, Christopher

Chemoproteomics validates selective targeting of Plasmodium M1 alanyl aminopeptidase as an antimalarial strategy

化学蛋白质组学验证了选择性靶向疟原虫 M1 丙氨酰氨基肽酶作为抗疟策略

Carlo Giannangelo #, Matthew P Challis #, Ghizal Siddiqui, Rebecca Edgar, Tess R Malcolm, Chaille T Webb, Nyssa Drinkwater, Natalie Vinh, Christopher Macraild, Natalie Counihan, Sandra Duffy, Sergio Wittlin, Shane M Devine, Vicky M Avery, Tania De Koning-Ward, Peter Scammells, Sheena McGowan, Darren

On-target, dual aminopeptidase inhibition provides cross-species antimalarial activity

靶向双氨基肽酶抑制提供跨物种抗疟活性

Rebecca C S Edgar, Tess R Malcolm, Ghizal Siddiqui, Carlo Giannangelo, Natalie A Counihan, Matthew Challis, Sandra Duffy, Mrittika Chowdhury, Jutta Marfurt, Madeline Dans, Grennady Wirjanata, Rintis Noviyanti, Kajal Daware, Chathura D Suraweera, Ric N Price, Sergio Wittlin, Vicky M Avery, Nyssa Drin

Promising antimalarial hits from phenotypic screens: a review of recently-described multi-stage actives and their modes of action

表型筛选中发现的有前景的抗疟药物:近期报道的多阶段活性成分及其作用机制综述

Luo, Annie-Peiyuan; Giannangelo, Carlo; Siddiqui, Ghizal; Creek, Darren J

Seasonality and Objective Physical Activity and Sedentary Behaviour among Older Adults from Four European Countries

来自四个欧洲国家的老年人的季节性、客观身体活动和久坐行为

Martins, João; Masoumi, Houshmand; Loureiro, Vânia; Gomes, Margarida; Ratinho, Fortunata; Ribeiro, Tiago; Mehriar, Melika; Rakovac, Marija; Šentija, Davor; Bahr, Andrzej; Tomczyk, Marta; Dynowski, Wojciech; Solinas, Roberto; Pirina, Maria Grazia; Coradduzza, Donatella; Boccuzzi, Giannangelo; Çağan, Birol; Dalcı, Ahmet; Papageorgiou, Athanasios; Smaga, Soultana; Parisopoulos, Georgios; Patsakas, Georgios; Meimaridis, Ioannis; Loureiro, Nuno; Marques, Adilson