日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Structure-Based Discovery of Hsp90/HDAC6 Dual Inhibitors Targeting Aggressive Prostate Cancer.

基于结构的Hsp90/HDAC6双重抑制剂的发现及其在侵袭性前列腺癌中的应用

Citarella Andrea, Belluti Silvia, Bonanni Davide, Moi Davide, Piccinini Isabella, Rinaldi Arianna, Papulino Chiara, Benedetti Rosaria, Cuoghi Laura, Ciolo Stefano Di, Silvani Alessandra, Altucci Lucia, Pinzi Luca, Franchini Silvia, Passarella Daniele, Sorbi Claudia, Giannini Clelia, Imbriano Carol, Rastelli Giulio

Combining Cyclic Triimidazo Triazine Core With Ethynyl-N-Methyl-Pyridinium Groups for Targeting G-Quadruplex Structures

将环状三咪唑三嗪核心与乙炔基-N-甲基吡啶鎓基团结合,用于靶向G-四链体结构

Platella, Chiara; Di Ciolo, Stefano; Criscuolo, Andrea; Malpicci, Daniele; Gaglione, Rosa; Arciello, Angela; Musumeci, Domenica; Lucenti, Elena; Cariati, Elena; Montesarchio, Daniela; Giannini, Clelia

Discovery of a Novel Trifluoromethyl Diazirine Inhibitor of SARS-CoV-2 M(pro)

发现一种新型三氟甲基重氮丙烯类SARS-CoV-2 M(pro)抑制剂

Citarella, Andrea; Moi, Davide; Pedrini, Martina; Pérez-Peña, Helena; Pieraccini, Stefano; Stagno, Claudio; Micale, Nicola; Schirmeister, Tanja; Sibille, Giulia; Gribaudo, Giorgio; Silvani, Alessandra; Passarella, Daniele; Giannini, Clelia

Novel Small Multilamellar Liposomes Containing Large Quantities of Peptide Nucleic Acid Selectively Kill Breast Cancer Cells

含有大量肽核酸的新型小型多层脂质体可选择性地杀死乳腺癌细胞

Proshkina, Galina; Shramova, Elena; Ryabova, Anastasiya; Katrivas, Liat; Giannini, Clelia; Malpicci, Daniele; Levi-Kalisman, Yael; Deyev, Sergey; Kotlyar, Alexander

Prompt and Long-Lived Anti-Kasha Emission from Organic Dyes

有机染料的快速持久抗卡沙排放

Malpicci, Daniele; Lucenti, Elena; Giannini, Clelia; Forni, Alessandra; Botta, Chiara; Cariati, Elena

Solid State Room Temperature Dual Phosphorescence from 3-(2-Fluoropyridin-4-yl)triimidazo[1,2-a:1',2'-c:1″,2″-e][1,3,5]triazine

3-(2-氟吡啶-4-基)三咪唑并[1,2-a:1',2'-c:1″,2″-e][1,3,5]三嗪的固态室温双重磷光

Previtali, Andrea; Lucenti, Elena; Forni, Alessandra; Mauri, Luca; Botta, Chiara; Giannini, Clelia; Malpicci, Daniele; Marinotto, Daniele; Righetto, Stefania; Cariati, Elena

The N-terminus of mature human frataxin is intrinsically unfolded

成熟人类弗拉塔辛蛋白的N端本身就是未折叠的。

Prischi, Filippo; Giannini, Clelia; Adinolfi, Salvatore; Pastore, Annalisa