日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Advancing Covalent Ligand and Drug Discovery beyond Cysteine

推进半胱氨酸以外的共价配体和药物发现

Kim, Gibae; Grams, R Justin; Hsu, Ku-Lung

Design, Synthesis, and Biological Evaluation of 5',7-Disubstituted 7-Deaza-adenosine Analogues as Irreversible Pan-FGFR Inhibitors

5',7-二取代7-脱氮腺苷类似物作为不可逆泛FGFR抑制剂的设计、合成和生物学评价

Park, Jung Hoon; Tran, Phuong Thao; Ko, Hye Lin; Mun, Seonghee; Jang, Sung Chul; Moon, Dong Hyun; Han, Jaeho; Kim, Jieun; Kim, Gibae; Choi, Hongseok; Kim, Seung Woo; Kim, Minjae; Lee, Sang Kook; Han, Byung Woo; Kang, Keon Wook; Jeong, Lak Shin

Structure-Activity Relationship Analysis of 2-Aryl-8-alkynyl Adenine and Nucleoside Scaffolds as A(3) Adenosine Receptor Ligands

2-芳基-8-炔基腺嘌呤和核苷骨架作为A(3)腺苷受体配体的构效关系分析

Kim, Gibae; Lee, Grim; Jarhad, Dnyandev B; Gao, Zhan-Guo; Kim, Seung Woo; Joung, Misuk; Jacobson, Kenneth A; Jeong, Lak Shin

Discovery of a Novel Template, N3‑1'-Homologated 4'-Truncated Thiosugar-Substituted Xanthine as an A(3)AR Antagonist via Conversion of an A(1)AR Antagonist

通过 A(1)AR 拮抗剂的转化,发现了一种新型模板,即 N3-1'-同系化的 4'-截短的硫代糖取代的黄嘌呤,作为 A(3)AR 拮抗剂。

Joung, Misuk; Kim, Minjae; Choi, Hongseok; Kim, Seung Woo; Kim, Gibae; Aswar, Vikas R; Baek, Seungwon; Kim, Hyun-Tae; Huh, Won-Ki; Jeong, Lak Shin

Design, Synthesis, and Biological Evaluation of C2-(N-Substituted Amino) Truncated 4'-Thioadenosine Derivatives as A(2A)AR and A(3)AR Dual Ligands

C2-(N-取代氨基)截短的4'-硫代腺苷衍生物作为A(2A)AR和A(3)AR双配体的设计、合成和生物学评价

Joung, Misuk; Choi, Hongseok; Kim, Minjae; Kim, Seung Woo; Kim, Gibae; Aswar, Vikas R; Baek, Seungwon; Kim, Hyun-Tae; Huh, Won-Ki; Jeong, Lak Shin

Comparative analysis of LJ-4378 and tirzepatide in mouse models of obesity and weight regain

LJ-4378 和 tirzepatide 在小鼠肥胖和体重反弹模型中的比较分析

Heeseong Kim # ,Seung Woo Kim # ,Cheoljun Choi ,SungUg Joo ,Gibae Kim ,Minjae Kim ,Eunsuk Yang ,Jangwon Lee ,Sukjae Chung ,Lak Shin Jeong ,Yun-Hee Lee

A Covalent PFKL Activator Suppresses Tumor Growth

共价PFKL激活剂抑制肿瘤生长

Jiang, Xiaoding; Lynch, Eric M; Lyu, Congcong; Wilson, Crystal; Salay, Lauren E; Lyons, Scott; Lu, Mu-Jie; Luo, Shuangyu; Kim, Gibae; Chan, Hsin-Ru; Wolfe, Wes; Lin, Yi-Chih; Kollman, Justin M; Cambronne, Xiaolu A; Hsu, Ku-Lung

Structure-Activity Relationship of Truncated 2,8-Disubstituted-Adenosine Derivatives as Dual A(2A)/A(3) Adenosine Receptor Antagonists and Their Cancer Immunotherapeutic Activity.

截短的 2,8-二取代腺苷衍生物作为双重 A(2A)/A(3) 腺苷受体拮抗剂的构效关系及其癌症免疫治疗活性

Kim Gibae, Hou Xiyan, Byun Woong Sub, Kim Gyudong, Jarhad Dnyandev B, Lee Grim, Hyun Young Eum, Yu Jinha, Lee Chang Soo, Qu Shuhao, Warnick Eugene, Gao Zhan-Guo, Kim Ji Yong, Ji Seunghee, Shin Hyunwoo, Choi Jong-Ryoul, Jacobson Kenneth A, Lee Hyuk Woo, Lee Sang Kook, Jeong Lak Shin

Discovery of a Novel Template, 7-Substituted 7-Deaza-4'-Thioadenosine Derivatives as Multi-Kinase Inhibitors

发现一种新型模板化合物,7-取代的7-脱氮-4'-硫代腺苷衍生物作为多激酶抑制剂

Mashelkar, Karishma K; Byun, Woong Sub; Ko, Hyejin; Sung, Kisu; Tripathi, Sushil K; An, Seungchan; Yum, Yun A; Kwon, Jee Youn; Kim, Minjae; Kim, Gibae; Kwon, Eun-Ji; Lee, Hyuk Woo; Noh, Minsoo; Lee, Sang Kook; Jeong, Lak Shin