日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Rational modulation of immune mechanisms synergizes the anti-tumor effects of targeted radiation therapy in pre-clinical models

在临床前模型中,合理调节免疫机制可增强靶向放射疗法的抗肿瘤作用。

Wirtz, Tristan; Lee, Catherine; Ram, Sripad; Xie, Tao; Mojtahedzadeh, Sepideh; Streiner, Nicole; Noorbehesht, Kavon; Manzuk, Lisa K; Rohner, Allison; Cabral, Edward; Bonato, Vinicius; Affolter, Timothy; Kraus, Manfred; Dillon, Christopher; Giddabasappa, Anand

18F-FLT PET, a Noninvasive Pharmacodynamic Biomarker of Tumor Cell Proliferation, Detected Differential Response to Various Cyclin-Dependent Kinase (CDK) Inhibitors

18F-FLT PET 是一种非侵入性的肿瘤细胞增殖药效学生物标志物,可检测到对各种细胞周期蛋白依赖性激酶 (CDK) 抑制剂的不同反应。

Giddabasappa, Anand; Jiang, Ziyue Karen; Yang, Bing; Chen, Laigao; Liu, Feng; Cabral, Edward; Ram, Sripad; Boras, Britton; Huser, Nanni; Zhang, Cathy C; Noorbehesht, Kavon; Manzuk, Lisa K; Visswanathan, Ravi; Mojtahedzadeh, Sepideh; Affolter, Timothy; Carmody, Jason; Kang, Aubrey Nayeon; Petroski, Matthew D; Khamphavong, Penny Lai; VanArsdale, Todd; Nguyen, Quang-Dé; Maresca, Kevin P; Dann, Stephen G

A Novel B7-H4xCD3 Bispecific T-cell Engager (PF-07260437) Synergizes with Breast Cancer Standard of Care and Immune Checkpoint Therapies

一种新型B7-H4xCD3双特异性T细胞衔接器(PF-07260437)与乳腺癌标准疗法和免疫检查点疗法具有协同作用

Keith Abayasiriwardana # ,Lei Wu # ,Hanane Laklai # ,Malgorzata Nocula-Lugowska ,Lioudmila Tchistiakova ,Jatin Narula ,Amy Jackson-Fisher ,Jonathon Golas ,My-Hanh Lam ,Veronika Grinstein ,Jung Wook Kang ,Jessica C Kearney ,Christine Hosselet ,Erik Upeslacis ,LuAnna Lemon ,Yun Zhang ,Changhua Ji ,Bernard S Buetow ,Martin B Finkelstein ,Netonia Marshall ,Stephanie Bisulco ,Edward Rosfjord ,Divya Mathur ,Jennifer Athanacio ,Ashley Thomas ,Alexander Trageser ,Diane Fernandez ,Ziyue Karen Jiang ,Sripad Ram ,Edward Cabral ,Lisa Manzuk ,Kevin Maresca ,Anand Giddabasappa ,Clare Lees ,Andrea T Hooper ,Puja Sapra ,Sudhakar Chintharlapalli

Advancing In Vivo Detection of T-Cell Function: Development and Preclinical Evaluation of (89)Zr-Ivuxolimab, a Human OX40 PET Tracer

推进体内T细胞功能检测:(89)Zr-Ivuxolimab(一种人源OX40 PET示踪剂)的开发和临床前评估

Kalita, Mausam; Kuo, Renesmee C; Reyes, Samantha T; Colburg, Deana Rae Crystal; Falk, Irene N; Anders, David; Vermesh, Ophir; Hayee, Samira; Azevedo, E Carmen; Nagy, Sydney C; Deal, Emily M; Chen, Anthony An-Fa Dahm; Kong, Christina S; Simonetta, Federico; Giddabasappa, Anand; Keliher, Edmund J; Bartlett, Derek W; Maresca, Kevin P; James, Michelle L; Alam, Israt S

Type I interferon regulation by USP18 is a key vulnerability in cancer

USP18 对 I 型干扰素的调控是癌症中的一个关键弱点。

Veronica Jové,Heather Wheeler,Chiachin Wilson Lee,David R Healy,Kymberly Levine,Erik C Ralph,Masaya Yamaguchi,Ziyue Karen Jiang,Edward Cabral,Yingrong Xu,Jeffrey Stock,Bing Yang,Anand Giddabasappa,Paula Loria,Agustin Casimiro-Garcia,Benedikt M Kessler,Adán Pinto-Fernández,Véronique Frattini,Paul D Wes,Feng Wang

Efficacy and Imaging-Enabled Pharmacodynamic Profiling of KRAS G12C Inhibitors in Xenograft and Genetically Engineered Mouse Models of Cancer

KRAS G12C抑制剂在异种移植和基因工程小鼠癌症模型中的疗效及影像辅助药效学分析

Lee, Catherine; Jiang, Ziyue Karen; Planken, Simon; Manzuk, Lisa K; Ortiz, Roberto; Hall, Michael; Noorbehesht, Kavon; Ram, Sripad; Affolter, Timothy; Troche, Gabriel E; Ihle, Nathan T; Johnson, Theodore; Ahn, Youngwook; Kraus, Manfred; Giddabasappa, Anand

Integrin αvβ8 on T cells suppresses anti-tumor immunity in multiple models and is a promising target for tumor immunotherapy

T细胞上的整合素αvβ8在多种模型中抑制抗肿瘤免疫,是肿瘤免疫治疗的一个有前景的靶点。

Eswari Dodagatta-Marri ,Hsiao-Yen Ma ,Benjia Liang ,John Li ,Dominique S Meyer ,Szu-Ying Chen ,Kai-Hui Sun ,Xin Ren ,Bahar Zivak ,Michael D Rosenblum ,Mark B Headley ,Lauren Pinzas ,Nilgun I Reed ,Joselyn S Del Cid ,Byron C Hann ,Sharon Yang ,Anand Giddabasappa ,Kavon Noorbehesht ,Bing Yang ,Joseph Dal Porto ,Tatsuya Tsukui ,Kyle Niessen ,Amha Atakilit ,Rosemary J Akhurst ,Dean Sheppard

Targeting and pharmacology of an anti-IL13Rα2 antibody and antibody-drug conjugate in a melanoma xenograft model

抗 IL13Rα2 抗体和抗体-药物偶联物在黑色素瘤异种移植模型中的靶向性和药理学

Parul Gupta, Ziyue Karen Jiang, Bing Yang, Lisa Manzuk, Edward Rosfjord, Johnny Yao, Luanna Lemon, Kavon Noorbehesht, John David, Sujiet Puthenveetil, Jeffrey M Casavant, Elwira Muszynska, Fengping Li, Mauricio Leal, Puja Sapra, Anand Giddabasappa

Preclinical Evaluation of 89Zr-Df-IAB22M2C PET as an Imaging Biomarker for the Development of the GUCY2C-CD3 Bispecific PF-07062119 as a T Cell Engaging Therapy

89Zr-Df-IAB22M2C PET 作为 GUCY2C-CD3 双特异性 PF-07062119 开发为 T 细胞接合疗法的影像生物标记物的临床前评估

Kevin P Maresca, Jianqing Chen, Divya Mathur, Anand Giddabasappa, Adam Root, Jatin Narula, Lindsay King, David Schaer, Jonathan Golas, Keith Kobylarz, Edward Rosfjord, Edmund Keliher, Laigao Chen, Sripad Ram, Eve H Pickering, James S Hardwick, Paul A Rejto, Amira Hussein, Ohad Ilovich, Kevin Staton,

Automated monitoring of respiratory rate as a novel humane endpoint: A refinement in mouse metastatic lung cancer models

呼吸频率自动监测作为一种新型人道终点指标:小鼠转移性肺癌模型的改进

Winn, Caroline B; Hwang, Seo-Kyoung; Morin, Jeffrey; Bluette, Crystal T; Manickam, Balasubramanian; Jiang, Ziyue K; Giddabasappa, Anand; Liu, Chang-Ning; Matthews, Kristin