日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Structural insights into isoform-specific RAS-PI3Kα interactions and the role of RAS in PI3Kα activation.

从结构角度深入了解 RAS-PI3Kα 同工型特异性相互作用以及 RAS 在 PI3Kα 激活中的作用

Czyzyk Daniel, Yan Wupeng, Messing Simon, Gillette William, Tsuji Takashi, Yamaguchi Mitsuhiro, Furuzono Shinji, Turner David M, Esposito Dominic, Nissley Dwight V, McCormick Frank, Simanshu Dhirendra K

Blocking C-terminal processing of KRAS4b via a direct covalent attack on the CaaX-box cysteine.

通过对 CaaX 盒半胱氨酸进行直接共价攻击,阻断 KRAS4b 的 C 端加工

Maciag Anna E, Yang Yue, Sharma Alok K, Turner David M, DeHart Caroline J, Abdelkarim Hazem, Fan Lixin, Smith Brian P, Kumari Vandana, Dyba Marcin, Rigby Megan, Castillo Badillo Jean A, Adams Lauren, Fornelli Luca, Fox Stephen, Brafman Alla, Turbyville Thomas, Gillette William, Messing Simon, Agamasu Constance, Wolfe Andrew L, Gysin Stephan, Chan Albert H, Simanshu Dhirendra K, Esposito Dominic, Chertov Oleg, Stephen Andrew G, Arkin Michelle, Renslo Adam, Kelleher Neil L, Gaponenko Vadim, Lightstone Felice C, Nissley Dwight V, McCormick Frank

Biophysical and structural analysis of KRAS switch-II pocket inhibitors reveals allele-specific binding constraints

对KRAS开关II口袋抑制剂的生物物理和结构分析揭示了等位基因特异性结合限制。

Alexander, Patrick; Chan, Albert H; Rabara, Dana; Swain, Monalisa; Larsen, Erik K; Dyba, Marcin; Chertov, Oleg; Ashraf, Mariam; Champagne, Allison; Lin, Ken; Maciag, Anna; Gillette, William K; Nissley, Dwight V; McCormick, Frank; Simanshu, Dhirendra K; Stephen, Andrew G

Improved production of class I phosphatidylinositol 4,5-bisphosphate 3-kinase.

提高 I 类磷脂酰肌醇 4,5-二磷酸 3-激酶的产量

Messing Simon, Widmeyer Stephanie R T, Denson John-Paul, Mehalko Jennifer, Wall Vanessa E, Drew Matthew, Snead Kelly, Hong Min, Grose Carissa, Esposito Dominic, Gillette William

NMR (1)H, (13)C, and (15)N resonance assignments of the oncogenic Q61R variant of human NRAS in the active, GTP-bound conformation

人类 NRAS 致癌 Q61R 变体在活性 GTP 结合构象下的 NMR (1)H、(13)C 和 (15)N 共振归属

Sharma, Alok K; Tonelli, Marco; Dyba, Marcin; Gillette, William K; Esposito, Dominic; Nissley, Dwight V; McCormick, Frank; Maciag, Anna E

Author Correction: Membrane lipids drive formation of KRAS4b-RAF1 RBDCRD nanoclusters on the membrane

作者更正:膜脂驱动膜上KRAS4b-RAF1 RBDCRD纳米簇的形成

Shrestha, Rebika; Carpenter, Timothy S; Van, Que N; Agamasu, Constance; Tonelli, Marco; Aydin, Fikret; Chen, De; Gulten, Gulcin; Glosli, James N; López, Cesar A; Oppelstrup, Tomas; Neale, Chris; Gnanakaran, Sandrasegaram; Gillette, William K; Ingólfsson, Helgi I; Lightstone, Felice C; Stephen, Andrew G; Streitz, Frederick H; Nissley, Dwight V; Turbyville, Thomas J

Membrane lipids drive formation of KRAS4b-RAF1 RBDCRD nanoclusters on the membrane

膜脂驱动膜上KRAS4b-RAF1 RBDCRD纳米簇的形成

Shrestha, Rebika; Carpenter, Timothy S; Van, Que N; Agamasu, Constance; Tonelli, Marco; Aydin, Fikret; Chen, De; Gulten, Gulcin; Glosli, James N; López, Cesar A; Oppelstrup, Tomas; Neale, Chris; Gnanakaran, Sandrasegaram; Gillette, William K; Ingólfsson, Helgi I; Lightstone, Felice C; Stephen, Andrew G; Streitz, Frederick H; Nissley, Dwight V; Turbyville, Thomas J

Producing recombinant proteins in Vibrio natriegens

在海洋弧菌中生产重组蛋白

Smith, Matthew; Hernández, José Sánchez; Messing, Simon; Ramakrishnan, Nitya; Higgins, Brianna; Mehalko, Jennifer; Perkins, Shelley; Wall, Vanessa E; Grose, Carissa; Frank, Peter H; Cregger, Julia; Le, Phuong Vi; Johnson, Adam; Sherekar, Mukul; Pagonis, Morgan; Drew, Matt; Hong, Min; Widmeyer, Stephanie R T; Denson, John-Paul; Snead, Kelly; Poon, Ivy; Waybright, Timothy; Champagne, Allison; Esposito, Dominic; Jones, Jane; Taylor, Troy; Gillette, William

Natural Product Graveoline Modulates Kirsten Rat Sarcoma Viral Oncogene Homologue (KRAS) Membrane Association: Insights from Advanced Spectroscopic Studies

天然产物格拉维林调节Kirsten大鼠肉瘤病毒癌基因同源物(KRAS)的膜结合:来自高级光谱学研究的启示

Cornilescu, Gabriel; Bindu, Lakshman; Sternicki, Louise; Chao, Fa-An; Gillette, William K; Fer, Nicole; Colombus, John; Castillo, Jean; Bonilla, Pedro Andrade; Van, Que N; Larsen, Erik; Hong, Min; Burgan, William; Turbyville, Thomas; Nissley, Dwight V; Liu, Miaomiao; Quinn, Ronald; Jean-Francois, Frantz L

Adapting recombinant bacterial alkaline phosphatase for nucleotide exchange of small GTPases.

改造重组细菌碱性磷酸酶用于小GTP酶的核苷酸交换

Frank Peter H, Hong Min, Higgins Brianna, Perkins Shelley, Taylor Troy, Wall Vanessa E, Drew Matthew, Waybright Timothy, Gillette William, Esposito Dominic, Messing Simon