日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Novel Sulfonium Reagents for the Modular Synthesis of Spiro[2.3]Hexanes and Heteroatom-Containing Analogues: Synthesis, Application, and Evaluation as Bioisosteres

用于模块化合成螺[2.3]己烷及其含杂原子类似物的新型锍试剂:合成、应用及作为生物等排体的评价

Natho, Philipp; Vicenti, Annarita; Mastrolorito, Fabrizio; De Franco, Francesca; Walsh-Benn, Lee; Colella, Marco; Mesto, Ernesto; Schingaro, Emanuela; Nicolotti, Orazio; Gioiello, Antimo; Luisi, Renzo

Structure-Based Discovery of Obeticholic Acid Derivatives as Novel Farnesoid X Receptor Partial Agonists with Improved Selectivity and Reduced Off-Target Effects

基于结构的奥贝胆酸衍生物作为新型法尼醇X受体部分激动剂的发现,具有更高的选择性和更低的脱靶效应

Passeri, Daniela; Cerra, Bruno; Carotti, Andrea; Greco, Francesco; Piermarini, Sara; Colliva, Carolina; Liscio, Paride; De Franco, Francesca; Adorini, Luciano; Erickson, Mary Ruth; Pellicciari, Roberto; Gioiello, Antimo

Coordinator Leadership in the Relationship Between Burnout and Nurses' Intention to Leave: A Cross-Sectional Study

协调员领导力在护士职业倦怠与离职意愿关系中的作用:一项横断面研究

Zaghini, Francesco; Marti, Flavio; Gonzalez, Cesar Ivan Aviles; Lo Monaco, Marika; Bartoli, Davide; Figura, Mariachiara; Gioiello, Giovanni

Expanding the Scope of PROTACs: Opportunities and Challenges in Topical Delivery

拓展PROTAC的范围:专题递送的机遇与挑战

Gioiello, Laura; Di Martino, Rita Maria Concetta; Pirali, Tracey

Discovery and development of steroidal enzyme inhibitors as anti-cancer drugs: state-of-the-art and future perspectives

甾体酶抑制剂作为抗癌药物的发现与开发:现状与展望

Cerra, Bruno; Gioiello, Antimo

Albuminuria is independently associated with preclinical left ventricular systolic dysfunction: The TESEO study

蛋白尿与临床前左心室收缩功能障碍独立相关:TESEO 研究

Barutta, Federica; Andreis, Alessandro; Bellettini, Matteo; Beccuti, Guglielmo; Ferro, Arianna; Bollati, Martina; Bellini, Stefania; Gioiello, Giulia; Mengozzi, Giulio; De Ferrari, Gaetano M; Alunni, Gianluca; Broglio, Fabio; Gruden, Gabriella

Comparison of Simoa and Lumipulse Neurofilament Light Chain Measurements in Alzheimer's Cerebrospinal Fluid: Preliminary Findings

Simoa 和 Lumipulse 检测阿尔茨海默病脑脊液中神经丝轻链的比较:初步研究结果

Boschi, Silvia; Chiarandon, Alberto Mario; Cermelli, Aurora; Lombardo, Chiara; Gioiello, Giulia; Montesano, Giulia; Rubino, Elisa; Mengozzi, Giulio; Rainero, Innocenzo; Roveta, Fausto

Ratiometric Two-Photon Near-Infrared Probe to Detect DPP IV in Human Plasma, Living Cells, Human Tissues, and Whole Organisms Using Zebrafish

使用比率双光子近红外探针检测斑马鱼中的人体血浆、活细胞、人体组织和整个生物体中的 DPP IV

Javier Valverde-Pozo, Jose M Paredes, Thomas J Widmann, Carmen Griñan-Lison, Giada Ceccarelli, Antimo Gioiello, M Eugenia Garcia-Rubiño, Juan A Marchal, Jose M Alvarez-Pez, Eva M Talavera

Multi-Gram Scale Synthesis and Characterization of Mometasone Furoate EP Impurity C

糠酸莫米松 EP 杂质 C 的克级合成与表征

Riccardo Ronchetti, Luigi Alfonso Pannone, Bruno Cerra, Emidio Camaioni, Gianfranco Lopopolo, Emanuele Attolino, Antimo Gioiello

Turning a Tumor Microenvironment Pitfall into Opportunity: Discovery of Benzamidoxime as PD-L1 Ligand with pH-Dependent Potency

将肿瘤微环境陷阱转化为机遇:发现苯甲酰胺肟作为具有 pH 依赖性效力的 PD-L1 配体

Elisa Bianconi, Alessandra Riccio, Luana Ruta, Carlo Bigiotti, Andrea Carotti, Sonia Moretti, Bruno Cerra, Antimo Gioiello, Simone Ferlin, Efisio Puxeddu, Antonio Macchiarulo