日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Exploiting the 2-(1,3,4,9-tetrahydropyrano[3,4-b]indol-1-yl)acetic Acid Scaffold to Generate COXTRANs: A New Class of Dual Cyclooxygenase Inhibitors-Thromboxane Receptor Antagonists

利用 2-(1,3,4,9-四氢吡喃并[3,4-b]吲哚-1-基)乙酸骨架生成 COXTRANs:一类新型双重环氧合酶抑制剂-血栓素受体拮抗剂

Blua, Federica; Boccato, Francesca; Buccellati, Carola; Risè, Patrizia; Barbieri, Silvia; Castiglioni, Laura; Balzulat, Annika; Rolando, Barbara; Marini, Elisabetta; Balestra, Marta; Introvigne, Maria Luisa; Giorgis, Marta; Sironi, Luigi; Tacconelli, Stefania; Hiesinger, Kerstin; Patrignani, Paola; Schmidtko, Achim; Steinhilber, Dieter; Proschak, Ewgenij; Sala, Angelo; Rovati, G Enrico; Bertinaria, Massimo

Fluorescent Isostere (Fluostere) of the Carboxylate: Design of hDHODH Fluorescent Inhibitors as Proof of Concept

羧酸盐的荧光等排体(Fluostere):hDHODH荧光抑制剂的设计及其概念验证

Sainas, Stefano; Martino, Elena; Garino, Claudio; Circosta, Paola; Luganini, Anna; Giorgis, Marta; Bavo, Francesco; Piccinini, Marco; Ramondetti, Cristina; Alberti, Marta; Miggiano, Riccardo; Gribaudo, Giorgio; Boschi, Donatella; Frølund, Bente; Lolli, Marco Lucio

Off-Target Inhibition of Human Dihydroorotate Dehydrogenase (hDHODH) Highlights Challenges in the Development of Fat Mass and Obesity-Associated Protein (FTO) Inhibitors.

人类二氢乳清酸脱氢酶 (hDHODH) 的脱靶抑制凸显了脂肪量和肥胖相关蛋白 (FTO) 抑制剂开发中的挑战

Tarullo Marco, Fernandez Rodriguez Guillermo, Iaiza Alessia, Venezia Sara, Macone Alberto, Incocciati Alessio, Masciarelli Silvia, Marchioni Marcella, Giorgis Marta, Lolli Marco Lucio, Fornaseri Federico, Proietti Ludovica, Grebien Florian, Rosignoli Serena, Paiardini Alessandro, Rotili Dante, Mai Antonello, Bochenkova Elena, Caflisch Amedeo, Fazi Francesco, Fatica Alessandro

Multitarget Antioxidant NO-Donor Organic Nitrates: A Novel Approach to Overcome Nitrates Tolerance, an Ex Vivo Study

多靶点抗氧化剂NO供体有机硝酸盐:克服硝酸盐耐受性的新方法——一项离体研究

Marini, Elisabetta; Giorgis, Marta; Leporati, Marta; Rolando, Barbara; Chegaev, Konstantin; Lazzarato, Loretta; Bertinaria, Massimo; Vincenti, Marco; Di Stilo, Antonella

A Comparative Study on the Efficacy of NLRP3 Inflammasome Signaling Inhibitors in a Pre-clinical Model of Bowel Inflammation

NLRP3炎症小体信号抑制剂在肠道炎症临床前模型中的疗效比较研究

Pellegrini, Carolina; Fornai, Matteo; Colucci, Rocchina; Benvenuti, Laura; D’Antongiovanni, Vanessa; Natale, Gianfranco; Fulceri, Federica; Giorgis, Marta; Marini, Elisabetta; Gastaldi, Simone; Bertinaria, Massimo; Blandizzi, Corrado; Antonioli, Luca