Discovery of cell active macrocyclic peptides with on-target inhibition of KRAS signaling
发现具有靶向抑制KRAS信号通路活性的细胞活性大环肽
期刊:Chemical Science
影响因子:7.4
doi:10.1039/d1sc05187c
Lim, Shuhui; Boyer, Nicolas; Boo, Nicole; Huang, Chunhui; Venkatachalam, Gireedhar; Angela Juang, Yu-Chi; Garrigou, Michael; Kaan, Hung Yi Kristal; Duggal, Ruchia; Peh, Khong Ming; Sadruddin, Ahmad; Gopal, Pooja; Yuen, Tsz Ying; Ng, Simon; Kannan, Srinivasaraghavan; Brown, Christopher J; Verma, Chandra S; Orth, Peter; Peier, Andrea; Ge, Lan; Yu, Xiang; Bhatt, Bhavana; Chen, Feifei; Wang, Erjia; Li, Nianyu Jason; Gonzales, Raymond J; Stoeck, Alexander; Henry, Brian; Sawyer, Tomi K; Lane, David P; Johannes, Charles W; Biswas, Kaustav; Partridge, Anthony W