日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A STAT3 degrader demonstrates efficacy in venetoclax resistant acute myeloid leukemia

STAT3降解剂在维奈托克耐药的急性髓系白血病中显示出疗效

Chakraborty, Samarpana; Morganti, Claudia; Zaldana, Kimberly; Rivera Pena, Bianca; Zhang, Hui; Verma, Divij; Gitego, Nadege; Ma, Feiyang; Aluri, Srinivas; Pradhan, Kith; Gordon-Mitchell, Shanisha; Mantzaris, Ioannis; Goldfinger, Mendel; Feldman, Eric; Gritsman, Kira; Shi, Yang; Hubner, Stefan; Qiu, Yi Hua; Brown, Brandon D; Khasawneh, Abdullah; Skwarska, Anna; de Camargo Magalhães, Eduardo Sabino; Verma, Amit; Konopleva, Marina; Tabe, Yoko; Gavathiotis, Evripidis; Colla, Simona; Gollob, Jared; Dey, Joyoti; Kornblau, Steven M; Koralov, Sergei B; Ito, Keisuke; Shastri, Aditi

Chemical modulation of cytosolic BAX homodimer potentiates BAX activation and apoptosis

细胞浆 BAX 同型二聚体的化学调节增强 BAX 活化和细胞凋亡

Nadege Gitego, Bogos Agianian, Oi Wei Mak, Vasantha Kumar Mv, Emily H Cheng, Evripidis Gavathiotis

Co-targeting of BAX and BCL-XL proteins broadly overcomes resistance to apoptosis in cancer

BAX 和 BCL-XL 蛋白的共同靶向广泛克服了癌症对细胞凋亡的抵抗

Andrea Lopez #, Denis E Reyna #, Nadege Gitego, Felix Kopp, Hua Zhou, Miguel A Miranda-Roman, Lars Ulrik Nordstrøm, Swathi-Rao Narayanagari, Ping Chi, Eduardo Vilar, Aristotelis Tsirigos, Evripidis Gavathiotis

ASXL1 mutations are associated with distinct epigenomic alterations that lead to sensitivity to venetoclax and azacytidine

ASXL1 突变与导致对维奈克拉和氮杂胞苷敏感性的明显表观基因组改变有关

Nora E Rahmani, Nandini Ramachandra, Srabani Sahu, Nadege Gitego, Andrea Lopez, Kith Pradhan, Tushar D Bhagat, Shanisha Gordon-Mitchell, Bianca Rivera Pena, Mohammad Kazemi, Keshav Rao, Orsi Giricz, Shahina Bano Maqbool, Raul Olea, Yongmei Zhao, Jinghang Zhang, Hamid Dolatshad, Vickram Tittrea, Dhar

Inhibitors of BRAF dimers using an allosteric site

使用变构位点的 BRAF 二聚体抑制剂

Xiomaris M Cotto-Rios #, Bogos Agianian #, Nadege Gitego, Emmanouil Zacharioudakis, Orsi Giricz, Yang Wu, Yiyu Zou, Amit Verma, Poulikos I Poulikakos, Evripidis Gavathiotis

Environment Dictates Dependence on Mitochondrial Complex I for NAD+ and Aspartate Production and Determines Cancer Cell Sensitivity to Metformin

环境决定了癌细胞对线粒体复合物 I 的依赖性,进而影响其对二甲双胍的敏感性。

Gui, Dan Y; Sullivan, Lucas B; Luengo, Alba; Hosios, Aaron M; Bush, Lauren N; Gitego, Nadege; Davidson, Shawn M; Freinkman, Elizaveta; Thomas, Craig J; Vander Heiden, Matthew G