日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Characterizing the binding of TC-5619 and encenicline on the alpha7 nicotinic acetylcholine receptor using PET imaging in the pig

使用 PET 成像在猪体内表征 TC-5619 和 encenicline 与 alpha7 烟碱乙酰胆碱受体的结合

Janus H Magnussen, Anders Ettrup, Szabolcs Lehel, Dan Peters, Agnete Dyssegaard, Morten S Thomsen, Jens D Mikkelsen, Gitte M Knudsen

Glucagon-like peptide-1 receptor regulation of basal dopamine transporter activity is species-dependent

胰高血糖素样肽-1受体对基础多巴胺转运体活性的调节具有物种依赖性

Mathias E Jensen, Aurelio Galli, Morgane Thomsen, Kathrine L Jensen, Gerda K Thomsen, Mette K Klausen, Tina Vilsbøll, Mikkel B Christensen, Jens J Holst, Anthony Owens, Sabrina Robertson, Lynette Daws, Daniele Zanella, Ulrik Gether, Gitte M Knudsen, Anders Fink-Jensen2

In Vitro and In Vivo Characterization of Dibenzothiophene Derivatives [125I]Iodo-ASEM and [18F]ASEM as Radiotracers of Homo- and Heteromeric α7 Nicotinic Acetylcholine Receptors

二苯并噻吩衍生物 [125I]碘-ASEM 和 [18F]ASEM 作为同源和异源 α7 烟碱乙酰胆碱受体放射性示踪剂的体外和体内表征

Cornelius K Donat, Henrik H Hansen, Hanne D Hansen, Ronnie C Mease, Andrew G Horti, Martin G Pomper, Elina T L'Estrade, Matthias M Herth, Dan Peters, Gitte M Knudsen, Jens D Mikkelsen

Blocking of efflux transporters in rats improves translational validation of brain radioligands

阻断大鼠的外排转运蛋白可改善脑放射性配体的转化验证

Vladimir Shalgunov, Mengfei Xiong, Elina T L'Estrade, Nakul R Raval, Ida V Andersen, Fraser G Edgar, Nikolaj R Speth, Simone L Baerentzen, Hanne D Hansen, Lene L Donovan, Arafat Nasser, Siv T Peitersen, Andreas Kjaer, Gitte M Knudsen, Stina Syvänen, Mikael Palner, Matthias M Herth

Synthesis and Pharmacological Evaluation of [11C]4-Methoxy- N-[2-(thiophen-2-yl)imidazo[1,2- a]pyridin-3-yl]benzamide as a Brain Penetrant PET Ligand Selective for the δ-Subunit-Containing γ-Aminobutyric Acid Type A Receptors

[11C]4-甲氧基-N-[2-(噻吩-2-基)咪唑并[1,2-a]吡啶-3-基]苯甲酰胺作为选择性针对含δ亚基的γ-氨基丁酸A型受体的脑渗透性PET配体的合成及药理学评价

Elina T L'Estrade, Hanne D Hansen, Christina Falk-Petersen, Anne Haugaard, Nane Griem-Krey, Sascha Jung, Hartmut Lüddens, Tanja Schirmeister, Maria Erlandsson, Tomas Ohlsson, Gitte M Knudsen, Matthias M Herth, Petrine Wellendorph, Bente Frølund

The Influence of the Toxin/Antitoxin mazEF on Growth and Survival of Listeria monocytogenes under Stress

毒素/抗毒素 mazEF 对压力下单核细胞增生李斯特菌生长和存活的影响

Thomas D Curtis, Ippei Takeuchi, Lone Gram, Gitte M Knudsen

The Small Colony Variant of Listeria monocytogenes Is More Tolerant to Antibiotics and Has Altered Survival in RAW 264.7 Murine Macrophages

单核细胞增生李斯特菌小菌落变体对抗生素的耐受性更强,并改变了 RAW 264.7 小鼠巨噬细胞中的存活率

Thomas D Curtis, Lone Gram, Gitte M Knudsen

Cerebral 5-HT2A receptor binding, but not mGluR2, is increased in tryptophan hydroxylase 2 decrease-of-function mice

色氨酸羟化酶 2 功能减退小鼠的大脑 5-HT2A 受体结合增加,但 mGluR2 没有增加

Christinna V Jørgensen, Jacob P Jacobsen, Marc G Caron, Anders B Klein, Gitte M Knudsen, Jens D Mikkelsen

α4βδ GABA(A) receptors are high-affinity targets for γ-hydroxybutyric acid (GHB)

α4βδ GABA(A) 受体是 γ-羟基丁酸 (GHB) 的高亲和力靶点

Nathan Absalom, Laura F Eghorn, Inge S Villumsen, Nasiara Karim, Tina Bay, Jesper V Olsen, Gitte M Knudsen, Hans Bräuner-Osborne, Bente Frølund, Rasmus P Clausen, Mary Chebib, Petrine Wellendorph

Cerebral markers of the serotonergic system in rat models of obesity and after Roux-en-Y gastric bypass

肥胖大鼠模型和 Roux-en-Y 胃绕道手术后的血清素系统脑标志物

Cecilia Ratner, Anders Ettrup, Marco Bueter, Mette E Haahr, Valérie Compan, Carel W le Roux, Barry Levin, Henrik H Hansen, Gitte M Knudsen