日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Biomanufacturing in low Earth orbit: A paradigm shift

近地轨道生物制造:范式转变

Marotta, Davide; Ward, Noor; Bauer, Steven R; Hunsberger, Joshua; Stoudemire, Jana; Savin, Kenneth; Giulianotti, Marc; Jamieson, Catriona H M; Roberts, Donna; Roberts, Michael

Structure-activity relationship of pyrrolidine pentamine derivatives as inhibitors of the aminoglycoside 6'- N -acetyltransferase type Ib

吡咯烷五胺衍生物作为氨基糖苷6'-N-乙酰转移酶Ib型抑制剂的构效关系

Sklenicka, Jan; Tran, Tung; Ramirez, Maria S; Donow, Haley M; Magaña, Angel J; LaVoi, Travis; Mamun, Yasir; Chapagain, Prem; Santos, Radleigh; Pinilla, Clemencia; Giulianotti, Marc A; Tolmasky, Marcelo E

Restoring susceptibility to aminoglycosides: identifying small molecule inhibitors of enzymatic inactivation

恢复对氨基糖苷类抗生素的敏感性:鉴定酶失活的小分子抑制剂

Magaña, Angel J; Sklenicka, Jan; Pinilla, Clemencia; Giulianotti, Marc; Chapagain, Prem; Santos, Radleigh; Ramirez, Maria Soledad; Tolmasky, Marcelo E

Biomanufacturing in low Earth orbit for regenerative medicine

利用近地轨道生物制造技术进行再生医学研究

Sharma, Arun; Clemens, Rachel A; Garcia, Orquidea; Taylor, D Lansing; Wagner, Nicole L; Shepard, Kelly A; Gupta, Anjali; Malany, Siobhan; Grodzinsky, Alan J; Kearns-Jonker, Mary; Mair, Devin B; Kim, Deok-Ho; Roberts, Michael S; Loring, Jeanne F; Hu, Jianying; Warren, Lara E; Eenmaa, Sven; Bozada, Joe; Paljug, Eric; Roth, Mark; Taylor, Donald P; Rodrigue, Gary; Cantini, Patrick; Smith, Amelia W; Giulianotti, Marc A; Wagner, William R

Identification and characterization of an atypical Gαs-biased β(2)AR agonist that fails to evoke airway smooth muscle cell tachyphylaxis

鉴定和表征一种非典型Gαs偏向性β(2)肾上腺素能受体激动剂,该激动剂无法诱发气道平滑肌细胞快速耐受性

Kim, Donghwa; Tokmakova, Alina; Lujan, Lauren K; Strzelinski, Hannah R; Kim, Nicholas; Najari Beidokhti, Maliheh; Giulianotti, Marc A; Mafi, Amirhossein; Woo, Jung-A A; An, Steven S; Goddard, William A 3rd; Liggett, Stephen B

Discovery of Nanomolar Melanocortin-3 Receptor (MC3R)-Selective Small Molecule Pyrrolidine Bis-Cyclic Guanidine Agonist Compounds Via a High-Throughput "Unbiased" Screening Campaign

通过高通量“无偏”筛选活动发现纳摩尔级黑素皮质素-3受体(MC3R)选择性小分子吡咯烷双环胍激动剂化合物

Doering, Skye R; Freeman, Katie; Debevec, Ginamarie; Geer, Phaedra; Santos, Radleigh G; Lavoi, Travis M; Giulianotti, Marc A; Pinilla, Clemencia; Appel, Jon R; Houghten, Richard A; Ericson, Mark D; Haskell-Luevano, Carrie

A Novel Class of Common Docking Domain Inhibitors That Prevent ERK2 Activation and Substrate Phosphorylation

一类新型的常见对接结构域抑制剂,可阻止ERK2激活和底物磷酸化

Sammons, Rachel M; Perry, Nicole A; Li, Yangmei; Cho, Eun Jeong; Piserchio, Andrea; Zamora-Olivares, Diana P; Ghose, Ranajeet; Kaoud, Tamer S; Debevec, Ginamarie; Bartholomeusz, Chandra; Gurevich, Vsevolod V; Iverson, Tina M; Giulianotti, Marc; Houghten, Richard A; Dalby, Kevin N

Identification of a Novel Polyamine Scaffold With Potent Efflux Pump Inhibition Activity Toward Multi-Drug Resistant Bacterial Pathogens

鉴定一种对多重耐药细菌病原体具有强效外排泵抑制活性的新型多胺支架

Fleeman, Renee M; Debevec, Ginamarie; Antonen, Kirsten; Adams, Jessie L; Santos, Radleigh G; Welmaker, Gregory S; Houghten, Richard A; Giulianotti, Marc A; Shaw, Lindsey N

Differential regulation of alcohol taking and seeking by antagonism at α4β2 and α3β4 nAChRs

通过拮抗α4β2和α3β4 nAChRs来差异性调节酒精摄入和渴求

Cippitelli, Andrea; Brunori, Gloria; Schoch, Jennifer; Armishaw, Christopher J; Wu, Jinhua; Zaveri, Nurulain T; Giulianotti, Marc A; Welmaker, Gregory S; Toll, Lawrence

Small-Molecule Inhibitors Targeting Topoisomerase I as Novel Antituberculosis Agents

靶向拓扑异构酶I的小分子抑制剂作为新型抗结核药物

Sandhaus, Shayna; Annamalai, Thirunavukkarasu; Welmaker, Greg; Houghten, Richard A; Paz, Carlos; Garcia, Pamela K; Andres, Angelo; Narula, Gagandeep; Rodrigues Felix, Carolina; Geden, Sandra; Netherton, Mandy; Gupta, Rashmi; Rohde, Kyle H; Giulianotti, Marc A; Tse-Dinh, Yuk-Ching