日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Orally Bioavailable Cyclin A/B RxL Inhibitors: Optimization of a Novel Class of Macrocyclic Peptides That Target E2F-High and G1-S-Checkpoint-Compromised Cancers

口服生物利用度高的细胞周期蛋白A/B RxL抑制剂:针对E2F高表达和G1-S检查点受损癌症的新型大环肽的优化

Shapiro, Justin A; Dupper, Nathan J; Fraga-Walton, Breena; Bockus, Andrew T; Leung, Siegfried S F; Yang, Kai; Bhatt, Chinmay; DeMart, Megan K; Baldomero, Miguel P; Hernandez, Luis; Fung, Gabriel; Metobo, Sammy; Xie, Steven; Lent, Bryan M; Spellmeyer, David C; Luna, Joshua; Hoang, Dalena; Chand, Manesh; Gritsenko, Yuliana; Gleason, Catherine E; Hamkins-Indik, Frances; Zheng, Jie; Odeh, Ranya; Nosrati, Meisam; He, Daphne; Bambal, Ramesh; Cremin, Peadar; Fang, Jinshu; Levin, Bernard; Wang, Evelyn W; Evangelista, Marie; Earp, David; Kreatsoulas, Constantine; Singh, Rajinder; Garcia, Pablo D; Aggen, James B

Cyclin A/B RxL Macrocyclic Inhibitors to Treat Cancers with High E2F Activity

细胞周期蛋白A/B RxL大环抑制剂用于治疗具有高E2F活性的癌症

Singh, Shilpa; Gleason, Catherine E; Fang, Min; Laimon, Yasmin N; Khivansara, Vishal; Xie, Shanhai; Durmaz, Yavuz T; Sarkar, Aniruddha; Ngo, Kenneth; Savla, Varunika; Li, Yixiang; Abu-Remaileh, Muhannad; Li, Xinyue; Tuladhar, Bishma; Odeh, Ranya; Hamkins-Indik, Frances; He, Daphne; Membreno, Miles W; Nosrati, Meisam; Gushwa, Nathan N; Leung, Siegfried S F; Fraga-Walton, Breena; Hernandez, Luis; Baldomero, Miguel P; Lent, Bryan M; Spellmeyer, David; Luna, Joshua F; Hoang, Dalena; Gritsenko, Yuliana; Chand, Manesh; DeMart, Megan K; Metobo, Sammy; Bhatt, Chinmay; Shapiro, Justin A; Yang, Kai; Dupper, Nathan J; Bockus, Andrew T; Doench, John G; Aggen, James B; Liu, Li-Fen; Levin, Bernard; Wang, Evelyn W; Vendrell, Iolanda; Fischer, Roman; Kessler, Benedikt; Gokhale, Prafulla C; Signoretti, Sabina; Spektor, Alexander; Kreatsoulas, Constantine; Singh, Rajinder; Earp, David J; Garcia, Pablo D; Nijhawan, Deepak; Oser, Matthew G

Potassium acts through mTOR to regulate its own secretion

钾离子通过 mTOR 调节自身的分泌。

Sørensen, Mads Vaarby; Saha, Bidisha; Jensen, Iben Skov; Wu, Peng; Ayasse, Niklas; Gleason, Catherine E; Svendsen, Samuel Levi; Wang, Wen-Hui; Pearce, David

Non-invasive detection of divergent metabolic signals in insulin deficiency vs. insulin resistance in vivo

体内无创检测胰岛素缺乏与胰岛素抵抗中不同的代谢信号

Morze, Cornelius von; Allu, Prasanna K R; Chang, Gene Y; Marco-Rius, Irene; Milshteyn, Eugene; Wang, Zhen J; Ohliger, Michael A; Gleason, Catherine E; Kurhanewicz, John; Vigneron, Daniel B; Pearce, David

Polyubiquitin binding to optineurin is required for optimal activation of TANK-binding kinase 1 and production of interferon β.

多聚泛素与 optineurin 结合是 TANK 结合激酶 1 的最佳激活和干扰素 β 产生的必要条件

Gleason Catherine E, Ordureau Alban, Gourlay Robert, Arthur J Simon C, Cohen Philip