日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

The Role of Intrinsically Disordered Domains in Regulating G Protein-Coupled Receptor Signaling

固有无序结构域在调节G蛋白偶联受体信号传导中的作用

Xu, Jun; Qiu, Ruoyi; Garces, Alexander M; Hübner, Harald; Xu, Xinyu; Hao, Chengyu; Weikert, Dorothee; Gmeiner, Peter; Lerch, Michael T; Kobilka, Brian K

Large Library Docking for Polypharmacology

用于多药理学的大型库对接

Wu, Yujin; Vigneron, Seth; Braz, Joao; Srinivasan, Karthik; Fink, Elissa A; Huang, Xi-Ping; Xu, Xinyu; Huebner, Harald; Kim, Joseph Y; Wang, Jing; Pfeiffer, Tara; Sakamoto, Kensuke; Radchenko, Dmytro S; Rodriguiz, Ramona M; Moroz, Yurii S; Irwin, John J; Gmeiner, Peter; Billesboelle, Christian; Roth, Bryan L; Basbaum, Allan I; Manglik, Aashish; Wetsel, William C; Shoichet, Brian K

LNP-Mediated CF10 Delivery Selectively Enhances Potency to Colorectal Cancer Cells and Preserves the TS/Top1 Dual Targeting Mechanism.

LNP介导的CF10递送选择性地增强了对结直肠癌细胞的效力,并保留了TS/Top1双重靶向机制。

Sarkar Santu, Behl Akanksha, Gmeiner William H

Preclinical Evaluation of a Radiolabeled Anti-PSMA Dimeric Aptamer in a Murine Model of Human Prostate Cancer

在人前列腺癌小鼠模型中对放射性标记的抗PSMA二聚体适体进行临床前评估

Sinha, Akesh; Pandya, Darpan N; Eeka, Prabhakar; Boyacioglu, Olcay; Gmeiner, William H; Wadas, Thaddeus J

CF10 Displays Improved Synergy with Oxaliplatin in TP53-Null and Wild-Type CRC Cells from Increased Top1cc and Replication Stress.

CF10 在 TP53 缺失型和野生型 CRC 细胞中与奥沙利铂表现出增强的协同作用,这是由于 Top1cc 增加和复制压力所致。

Young Taylor M, Moumouni Rida, Behl Akanksha, Das Upasana, Gmeiner William H

Using causal machine learning and real world data to improve dose response decision making for secukinumab in psoriatic arthritis

利用因果机器学习和真实世界数据改进司库奇尤单抗治疗银屑病关节炎的剂量反应决策

Kiltz, Uta; Glassen, Thomas; Brandt-Juergens, Jan; Kiss, Ferenc; Peterlik, Daniel; Gmeiner, Benjamin

Testing a digitally administered intervention to increase social participation, physical fitness, and health awareness among healthy older adults by means of tablet-based app use: study protocol of the SMART-AGE randomized controlled trial

一项旨在通过平板电脑应用程序提高健康老年人社会参与度、身体素质和健康意识的数字化干预措施的测试:SMART-AGE随机对照试验的研究方案

Memmer, Nicole; Snijder-Steinhilber, Meike; Burkhardt, Heinrich; Hellmund, Claudia; Jansen, Carl-Philipp; Kölsch, Verena M; Krönung, Julia; Kuhlmann, Beatrice G; Masia, Lorenzo; Oswald, Frank; Paech, Barbara; Radeck, Leon; Schlomann, Anna; Schmidt, Laura I; Stefanakis, Marios E; Wanka, Anna; Kramer-Gmeiner, Franziska; Böttinger, Melissa; Ewert, Janina; Kniepkamp, Sophie; Gordt-Osterwind, Katharina; Litz, Elena; Mertens, Alica; Sperling, Uwe; Ehni, Hans-Jörg; Becker, Clemens; Wahl, Hans-Werner; Schubert, Anna-Lena; Eckert, Tobias; Bauer, Jürgen

The fluoropyrimidine polymer CF10 synergizes with 5-ethynyl-2'-deoxyuridine by promoting telomere attrition and mitotic catastrophe

氟嘧啶聚合物CF10与5-乙炔基-2'-脱氧尿苷协同作用,促进端粒损耗和有丝分裂灾难。

Das, Upasana; Behl, Akanksha; Gmeiner, William H

Synthesis and Characterization of Photoswitchable Covalent Ligands for the β(2)-Adrenoceptor

β(2)-肾上腺素受体光开关共价配体的合成与表征

Wirth, Ulrike; Neu, Eduard; Provasi, Davide; Feustel, Steffen; Schmidt, Maximilian F; Hübner, Harald; Weikert, Dorothée; Filizola, Marta; König, Burkhard; Gmeiner, Peter

Mechanism and function of GPR3 regulated by a negative allosteric modulator.

负变构调节剂调控 GPR3 的机制和功能

Chen Geng, Bláhová Jana, Staffen Nico, Hübner Harald, Nunhöfer Nadja, Qiu Chen, Gmeiner Peter, Weikert Dorothee, Du Yang, Xu Jun