日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

The Role of Intrinsically Disordered Domains in Regulating G Protein-Coupled Receptor Signaling

固有无序结构域在调节G蛋白偶联受体信号传导中的作用

Xu, Jun; Qiu, Ruoyi; Garces, Alexander M; Hübner, Harald; Xu, Xinyu; Hao, Chengyu; Weikert, Dorothee; Gmeiner, Peter; Lerch, Michael T; Kobilka, Brian K

Large Library Docking for Polypharmacology

用于多药理学的大型库对接

Wu, Yujin; Vigneron, Seth; Braz, Joao; Srinivasan, Karthik; Fink, Elissa A; Huang, Xi-Ping; Xu, Xinyu; Huebner, Harald; Kim, Joseph Y; Wang, Jing; Pfeiffer, Tara; Sakamoto, Kensuke; Radchenko, Dmytro S; Rodriguiz, Ramona M; Moroz, Yurii S; Irwin, John J; Gmeiner, Peter; Billesboelle, Christian; Roth, Bryan L; Basbaum, Allan I; Manglik, Aashish; Wetsel, William C; Shoichet, Brian K

Synthesis and Characterization of Photoswitchable Covalent Ligands for the β(2)-Adrenoceptor

β(2)-肾上腺素受体光开关共价配体的合成与表征

Wirth, Ulrike; Neu, Eduard; Provasi, Davide; Feustel, Steffen; Schmidt, Maximilian F; Hübner, Harald; Weikert, Dorothée; Filizola, Marta; König, Burkhard; Gmeiner, Peter

Mechanism and function of GPR3 regulated by a negative allosteric modulator.

负变构调节剂调控 GPR3 的机制和功能

Chen Geng, Bláhová Jana, Staffen Nico, Hübner Harald, Nunhöfer Nadja, Qiu Chen, Gmeiner Peter, Weikert Dorothee, Du Yang, Xu Jun

Discovery of a functionally selective serotonin receptor (5-HT(1A)R) agonist for the treatment of pain.

发现一种功能选择性血清素受体(5-HT(1A)R)激动剂用于治疗疼痛

Ullrich Annika, Schneider Johannes, Braz João M, Neu Eduard, Staffen Nico, Stanek Markus, Bláhová Jana, Hove Tamsanqa, Albert Tamara, Allikalt Anni, Löber Stefan, Bhardwaj Karnika, Rodriguez-Rosado Sian, Fink Elissa, Rasmussen Tim, Hübner Harald, Inoue Asuka, Shoichet Brian K, Basbaum Allan I, Böttcher Bettina, Weikert Dorothee, Gmeiner Peter

Acid sphingomyelinase activity suggests a new antipsychotic pharmaco-treatment strategy for schizophrenia

酸性鞘磷脂酶活性提示了一种治疗精神分裂症的新型抗精神病药物治疗策略

Chestnykh, Daria; Mühle, Christiane; Schumacher, Fabian; Kalinichenko, Liubov S; Löber, Stefan; Gmeiner, Peter; Alzheimer, Christian; von Hörsten, Stephan; Kleuser, Burkhard; Uebe, Steffen; Ekici, Arif B; Gulbins, Erich; Kornhuber, Johannes; Jin, Hee Kyung; Bae, Jae-Sung; Lourdusamy, Anbarasu; Müller, Christian P

(99m)Tc-Labeled Diarylpyrazoles for Single-Emission Computer Tomography Imaging of Neurotensin Receptor-Positive Tumors: A Comparative Preclinical Study

(99m)Tc标记的二芳基吡唑用于神经降压素受体阳性肿瘤的单发射计算机断层扫描成像:一项比较性临床前研究

Potemkin, Roman; Maschauer, Simone; Hübner, Harald; Kuwert, Torsten; Bäuerle, Tobias; Gmeiner, Peter; Prante, Olaf

SAG1.3-derived Frizzled-targeting small-molecule compounds.

源自 SAG1.3 的 Frizzled 靶向小分子化合物。

Grätz Lukas, Turku Ainoleena, Kozielewicz Pawel, Bowin Carl-Fredrik, Scharf Magdalena M, Voss Jan H, Kinsolving Julia, Shekhani Rawan, Oliva-Vilarnau Nuria, Koolmeister Tobias, Körber Marlies, Lauschke Volker M, Löber Stefan, Gmeiner Peter, Schulte Gunnar

The role of intrinsically disordered domains in regulating G protein coupled receptor signaling

固有无序结构域在调节G蛋白偶联受体信号传导中的作用

Xu, Jun; Qiu, Ruoyi; Garces, Alexander M; Hübner, Harald; Xu, Xinyu; Weikert, Dorothee; Gmeiner, Peter; Lerch, Michael T; Kobilka, Brian K

Structural and functional characterization of the endogenous agonist for orphan receptor GPR3

孤儿受体GPR3内源性激动剂的结构和功能表征

Chen, Geng; Staffen, Nico; Wu, Zhangsong; Xu, Xinyu; Pan, Jinheng; Inoue, Asuka; Shi, Tingyi; Gmeiner, Peter; Du, Yang; Xu, Jun