日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Restructuring Antiviral Quinazolinone Frameworks to Derive and Optimize Inhibitors of Chikungunya Virus

重构抗病毒喹唑啉酮骨架以衍生和优化基孔肯雅病毒抑制剂

Roach, Caroline M; Streblow, Zachary J; Zhang, Yuting; Ogorek, Tyler J; Ponce-Flores, Alejandro; Jonsson, Colleen B; Streblow, Daniel N; Golden, Jennifer E

Broad spectrum antiviral BDGR-164 provides protection against lethal neurotropic alphavirus infection in mice

广谱抗病毒药物BDGR-164可保护小鼠免受致命性嗜神经性甲病毒感染。

Williams, Evan P; Xue, Yi; Yang, Dong; Lee, Jasper; Kim, Eunjung; Ponce-Flores, Alexander; Zalduondo, Lillian; Cao, Xufeng; Chung, Donghoon; Golden, Jennifer E; Meibohm, Bernd; Fitzpatrick, Elizabeth A; Weaver, Scott C; Jonsson, Colleen B

The antiviral BDGR-49 provides protection from lethal, neurotropic Venezuelan equine encephalitis virus intranasal infection in mice.

抗病毒药物 BDGR-49 可保护小鼠免受致命的嗜神经性委内瑞拉马脑炎病毒鼻内感染

Williams Evan P, Xue Yi, Vogel Peter, Yang Dong, Ponce-Flores Alejandro, Li Xiaoyu, Ogorek Tyler J, Saini Manisha, Iulek Jorge, Ruiz Francesc Xavier, Arnold Eddy, Golden Jennifer E, Meibohm Bernd, Jonsson Colleen B

Pharmacophore Establishment and Optimization of Saturated 1,6-Naphthyridine-Fused Quinazolinones that Inhibit Meningoencephalitis-Causing Naegleria fowleri

抑制引起脑膜脑炎的福氏耐格里阿米巴的饱和1,6-萘啶稠合喹唑啉酮的药效团建立与优化

Lish, Matthew S; McKeon, Jillian E M; Palmentiero, Caroline M; Pomeroy, Julia M; Roster, Colm P; Guzei, Ilia A; Morris, James C; Golden, Jennifer E

Synthesis and Evaluation of Benzylamine Inhibitors of Neuropathogenic Naegleria fowleri "Brain-Eating" Amoeba

神经致病性福氏耐格里“食脑”变形虫苄胺抑制剂的合成与评价

Pomeroy, Julia M; Khalifa, Muhammad M; Milanes, Jillian E; Palmentiero, Caroline M; Morris, James C; Golden, Jennifer E

Efficacy of a brain-penetrant antiviral in lethal Venezuelan and eastern equine encephalitis mouse models

脑穿透性抗病毒药物在致命性委内瑞拉脑炎和东部马脑炎小鼠模型中的疗效

Cao, Xufeng; Yang, Dong; Parvathareddy, Jyothi; Chu, Yong-Kyu; Kim, Eun Jung; Fitz-Henley, Jhewelle N; Li, Xiaoyu; Lukka, Pradeep B; Parmar, Keyur R; Temrikar, Zaid H; Dhole, Priya; Adcock, Robert Scott; Gabbard, Jon; Bansal, Shruti; Lee, Jasper; Zalduondo, Lillian; Hayes, Ernestine; Stabenow, Jennifer; Meibohm, Bernd; Fitzpatrick, Elizabeth A; Bailey, Kevin; Campos, Rafael K; Julander, Justin G; Rossi, Shannan L; Chung, Donghoon; Jonsson, Colleen B; Golden, Jennifer E

Clinical and Translational Pharmacology Considerations for Anti-infectives Approved Under the FDA Animal Rule

根据FDA动物规则批准的抗感染药物的临床和转化药理学考量

Temrikar, Zaid H; Golden, Jennifer E; Jonsson, Colleen B; Meibohm, Bernd

Mannich-Type Condensation and Domino Quinazolinone-Amidine Rearrangement Affords Ring-Fused Mackinazolinones with Anti-Amoebic Activity

曼尼希型缩合和多米诺喹唑啉酮-脒重排反应生成具有抗阿米巴活性的稠环麦基唑啉酮。

Lish, Matthew S; Milanes, Jillian E; Sanders, Kyana M; Guzei, Ilia A; Morris, James C; Golden, Jennifer E

Advances in the Development of Small Molecule Antivirals against Equine Encephalitic Viruses

抗马脑炎病毒小分子抗病毒药物研发进展

Ogorek, Tyler J; Golden, Jennifer E

Characterization of Glucokinases from Pathogenic Free-Living Amoebae

致病性自由生活变形虫葡萄糖激酶的特性分析

Milanes, Jillian E; Suryadi, Jimmy; Monaghan, Neil P; Harding, Elijah M; Morris, Corbin S; Rozema, Soren D; Khalifa, Muhammad M; Golden, Jennifer E; Phan, Isabelle Q; Zigweid, Rachael; Abendroth, Jan; Rice, Christopher A; McCord, Hayden T; Wilson, Stevin; Fenwick, Michael K; Morris, James C