日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Second-site suppressor mutations reveal connection between the drug-binding pocket and nucleotide-binding domain 1 of human P-glycoprotein (ABCB1).

第二位点抑制突变揭示了人类 P-糖蛋白 (ABCB1) 的药物结合口袋与核苷酸结合域 1 之间的联系

Murakami Megumi, Sajid Andaleeb, Lusvarghi Sabrina, Durell Stewart R, Abel Biebele, Vahedi Shahrooz, Golin John, Ambudkar Suresh V

Abstract 1382: Visualization and functional annotation of coronavirus spike protein glycoshields

摘要 1382:冠状病毒刺突蛋白糖基化的可视化和功能注释

Alhumaidi, Maryam; Nentwig, Lea-Marie; Rahman, Hadiar; Schmitt, Lutz; Rudrow, Andrew; Harris, Andrzej; Dillon, Cierra; Restrepo, Lucas; Lamping, Erwin; Arya, Nidhi; Ambudkar, Suresh V; Choy, John S; Golin, John; Hsu, Shang-Te Danny; Yang, Tzu-Jing; Yu, Pei-Yu; Tsai, Yu-Xi; Chang, Ning-En; Khoo, Kay-Hooi; Hanus, Cyril; Sikora, Mateusz

Residues forming the gating regions of asymmetric multidrug transporter Pdr5 also play roles in conformational switching and protein folding

构成不对称多药转运蛋白Pdr5门控区域的残基也参与构象转换和蛋白质折叠。

Alhumaidi, Maryam; Nentwig, Lea-Marie; Rahman, Hadiar; Schmitt, Lutz; Rudrow, Andrew; Harris, Andrzej; Dillon, Cierra; Restrepo, Lucas; Lamping, Erwin; Arya, Nidhi; Ambudkar, Suresh V; Choy, John S; Golin, John

An A666G mutation in transmembrane helix 5 of the yeast multidrug transporter Pdr5 increases drug efflux by enhancing cooperativity between transport sites

酵母多药转运蛋白Pdr5跨膜螺旋5中的A666G突变通过增强转运位点之间的协同作用来增加药物外排。

Arya, Nidhi; Rahman, Hadiar; Rudrow, Andrew; Wagner, Manuel; Schmitt, Lutz; Ambudkar, Suresh V; Golin, John

Robust, pleiotropic drug resistance 5 (Pdr5)-mediated multidrug resistance is vigorously maintained in Saccharomyces cerevisiae cells during glucose and nitrogen limitation

在葡萄糖和氮限制条件下,酿酒酵母细胞中由Pdr5介导的强效、多效性耐药性得以维持。

Rahman, Hadiar; Carneglia, Joshua; Lausten, Molly; Robertello, Michael; Choy, John; Golin, John

The multidrug transporter Pdr5 on the 25th anniversary of its discovery: an important model for the study of asymmetric ABC transporters

多药转运蛋白Pdr5发现25周年:研究不对称ABC转运蛋白的重要模型

Golin, John; Ambudkar, Suresh V

Mutations define cross-talk between the N-terminal nucleotide-binding domain and transmembrane helix-2 of the yeast multidrug transporter Pdr5: possible conservation of a signaling interface for coupling ATP hydrolysis to drug transport

突变揭示了酵母多药转运蛋白Pdr5的N端核苷酸结合域与跨膜螺旋2之间的相互作用:可能存在一个保守的信号转导界面,用于将ATP水解与药物转运偶联起来。

Sauna, Zuben E; Bohn, Sherry Supernavage; Rutledge, Robert; Dougherty, Michael P; Cronin, Susan; May, Leopold; Xia, Di; Ambudkar, Suresh V; Golin, John