NBI-921352, a first-in-class, NaV1.6 selective, sodium channel inhibitor that prevents seizures in Scn8a gain-of-function mice, and wild-type mice and rats
NBI-921352 是一种首创的 NaV1.6 选择性钠通道抑制剂,可预防 Scn8a 功能获得小鼠以及野生型小鼠和大鼠的癫痫发作
期刊:Elife
影响因子:6.4
doi:10.7554/eLife.72468
J P Johnson, Thilo Focken, Kuldip Khakh, Parisa Karimi Tari, Celine Dube, Samuel J Goodchild, Jean-Christophe Andrez, Girish Bankar, David Bogucki, Kristen Burford, Elaine Chang, Sultan Chowdhury, Richard Dean, Gina de Boer, Shannon Decker, Christoph Dehnhardt, Mandy Feng, Wei Gong, Michael Grimwood