日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Synthesis of 2,3-dihydrobenzo[b][1,4]dioxine-5-carboxamide and 3-oxo-3,4-dihydrobenzo[b][1,4]oxazine-8-carboxamide derivatives as PARP1 inhibitors

2,3-二氢苯并[b][1,4]二氧杂环己烯-5-甲酰胺和3-氧代-3,4-二氢苯并[b][1,4]恶嗪-8-甲酰胺衍生物作为PARP1抑制剂的合成

Xuwei Shao, Steven Pak, Uday Kiran Velagapudi, Shruthi Gobbooru, Sai Shilpa Kommaraju, Woon-Kai Low, Gopal Subramaniam, Sanjai Kumar Pathak, Tanaji T Talele

Development of a highly potent, selective, and cell-active inhibitor of cysteine cathepsin L-A hybrid design approach

开发高效、选择性和细胞活性的半胱氨酸蛋白酶抑制剂 LA 混合设计方法

Dibyendu Dana, Shatarupa De, Pratikkumar Rathod, Anibal R Davalos, Daniel A Novoa, Suneeta Paroly, Viviana M Torres, Nisar Afzal, Ravi S Lankalapalli, Susan A Rotenberg, Emmanuel J Chang, Gopal Subramaniam, Sanjai Kumar

Development of cell-active non-peptidyl inhibitors of cysteine cathepsins

细胞活性非肽基半胱氨酸蛋白酶抑制剂的开发

Dibyendu Dana, Anibal R Davalos, Shatarupa De, Pratikkumar Rathod, Ranjith K Gamage, Juliana Huestis, Nisar Afzal, Yuriy Zavlanov, Suneeta S Paroly, Susan A Rotenberg, Gopal Subramaniam, Kevin J Mark, Emmanuel J Chang, Sanjai Kumar