日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Human aminolevulinate synthase structure reveals a eukaryotic-specific autoinhibitory loop regulating substrate binding and product release

人类氨基乙酰丙酸合酶结构揭示了真核生物特异性自抑制环路调节底物结合和产物释放

Henry J Bailey #, Gustavo A Bezerra #, Jason R Marcero #, Siladitya Padhi #, William R Foster, Elzbieta Rembeza, Arijit Roy, David F Bishop, Robert J Desnick, Gopalakrishnan Bulusu, Harry A Dailey Jr, Wyatt W Yue

2-[2-(4-(trifluoromethyl)phenylamino)thiazol-4-yl]acetic acid (Activator-3) is a potent activator of AMPK

2-[2-(4-(三氟甲基)苯氨基)噻唑-4-基]乙酸 (Activator-3) 是一种有效的 AMPK 激活剂

Navneet Bung, Sobhitha Surepalli, Sriram Seshadri, Sweta Patel, Saranya Peddasomayajula, Lalith Kumar Kummari, Sireesh T Kumar, Phanithi Prakash Babu, Kishore V L Parsa, Rajamohan Reddy Poondra, Gopalakrishnan Bulusu, Parimal Misra

A novel SIRT1 inhibitor, 4bb induces apoptosis in HCT116 human colon carcinoma cells partially by activating p53

新型 SIRT1 抑制剂 4bb 部分通过激活 p53 诱导 HCT116 人结肠癌细胞凋亡

Ananga Ghosh, Amrita Sengupta, Guru Pavan Kumar Seerapu, Ali Nakhi, E V Venkat Shivaji Ramarao, Navneet Bung, Gopalakrishnan Bulusu, Manojit Pal, Devyani Haldar