Novel Macrocyclic Antagonists of the CGRP Receptor Part 2: Stereochemical Inversion Induces an Unprecedented Binding Mode
CGRP受体的新型大环拮抗剂(第二部分):立体化学反转诱导了一种前所未有的结合模式
期刊:ACS Medicinal Chemistry Letters
影响因子:4
doi:10.1021/acsmedchemlett.2c00400
Southall, Stacey M; Banerjee, Joydeep; Brown, Jason; Butkovic, Kristina; Cansfield, Andrew D; Cansfield, Julie E; Congreve, Miles S; Cseke, Gabriella; Deflorian, Francesca; Hunjadi, Martina Petrovic; Hutinec, Antun; Inturi, Trinadh Kumar; Rupcic, Renata; Saxty, Gordon; Watson, Stephen P