日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

ADT-1004: a first-in-class, oral pan-RAS inhibitor with robust antitumor activity in preclinical models of pancreatic ductal adenocarcinoma

ADT-1004:一种首创的口服泛RAS抑制剂,在胰腺导管腺癌的临床前模型中具有强大的抗肿瘤活性

Bandi, Dhana Sekhar Reddy; Nagaraju, Ganji Purnachandra; Sarvesh, Sujith; Carstens, Julienne L; Foote, Jeremy B; Graff, Emily C; Fang, Yu-Hua D; Keeton, Adam B; Chen, Xi; Valiyaveettil, Jacob; Berry, Kristy L; Bae, Sejong; Akce, Mehmet; Gorman, Greg; Yoon, Karina J; Manne, Upender; Boyd, Michael R; Buchsbaum, Donald J; Azmi, Asfar S; Maxuitenko, Yulia Y; Piazza, Gary A; El-Rayes, Bassel F

A Pan-RAS Inhibitor with a Unique Mechanism of Action Blocks Tumor Growth and Induces Antitumor Immunity in Gastrointestinal Cancer.

一种具有独特作用机制的泛 RAS 抑制剂可抑制肿瘤生长并诱导胃肠道癌症的抗肿瘤免疫

Foote Jeremy B, Mattox Tyler E, Keeton Adam B, Chen Xi, Smith Forrest T, Berry Kristy, Holmes Thomas W, Wang Junwei, Huang Chung-Hui, Ward Antonio, Mitra Amit K, Ramirez-Alcantara Veronica, Hardy Cherlene, Fleten Karianne G, Flatmark Kjersti, Yoon Karina J, Sarvesh Sujith, Nagaraju Ganji P, Bandi Dhana Sekhar Reddy, Maxuitenko Yulia Y, Valiyaveettil Jacob, Carstens Julienne L, Buchsbaum Donald J, Yang Jennifer, Zhou Gang, Nurmemmedov Elmar, Babic Ivan, Gaponeko Vadim, Abdelkarim Hazem, Boyd Michael R, Gorman Greg, Manne Upender, Bae Sejong, El-Rayes Bassel F, Piazza Gary A

Multicenter Phase IB Trial of Carboxyamidotriazole Orotate and Temozolomide for Recurrent and Newly Diagnosed Glioblastoma and Other Anaplastic Gliomas

羧酰胺三唑乳清酸盐联合替莫唑胺治疗复发性和新诊断的胶质母细胞瘤及其他间变性胶质瘤的多中心IB期临床试验

Omuro, Antonio; Beal, Kathryn; McNeill, Katharine; Young, Robert J; Thomas, Alissa; Lin, Xuling; Terziev, Robert; Kaley, Thomas J; DeAngelis, Lisa M; Daras, Mariza; Gavrilovic, Igor T; Mellinghoff, Ingo; Diamond, Eli L; McKeown, Andrew; Manne, Malbora; Caterfino, Andrew; Patel, Krishna; Bavisotto, Linda; Gorman, Greg; Lamson, Michael; Gutin, Philip; Tabar, Viviane; Chakravarty, Debyani; Chan, Timothy A; Brennan, Cameron W; Garrett-Mayer, Elizabeth; Karmali, Rashida A; Pentsova, Elena

The TAM receptor Mertk protects against neuroinvasive viral infection by maintaining blood-brain barrier integrity

TAM 受体 Mertk 通过维持血脑屏障完整性来预防神经侵入性病毒感染

Jonathan J Miner, Brian P Daniels, Bimmi Shrestha, Jose L Proenca-Modena, Erin D Lew, Helen M Lazear, Matthew J Gorman, Greg Lemke, Robyn S Klein, Michael S Diamond

A novel and rapid LC/MS/MS assay for bioanalysis of Azurin p28 in serum and its pharmacokinetics in mice

一种新型快速的LC/MS/MS方法用于血清中Azurin p28的生物分析及其在小鼠体内的药代动力学研究。

Gorman, Greg S; Coward, Lori U; Freeman, Lea; Noker, Pat E; Beattie, Craig W; Jia, Lee