日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Proximity-Induced Rewiring of Oncogenic Kinase Triggers Apoptosis

邻近诱导的致癌激酶重编程触发细胞凋亡

Merz, Manuel L; Shoba, Veronika M; Pergu, Rajaiah; Severance, Zachary C; Munkanatta Godage, Dhanushka N P; Deb, Arghya; Kwok, Hui Si; Singh, Prashant; Singh, Sameek; Allen, Jonathan B; Tian, Wenzhi; Gosavi, Pallavi M; Chaudhary, Santosh K; Anokhina, Viktoriya; Weisberg, Ellen L; Payne, N Connor; He, Yao; Dhaliwal, Rohil; Osadchey, Reilly; Shekhar, Mrinal; Mazitschek, Ralph; Rees, Matthew G; Roth, Jennifer A; Cui, Qiang; Griffin, James D; Liau, Brian B; Choudhary, Amit

Phosphorylation-inducing chimera rewires oncogenic kinase to trigger apoptosis.

磷酸化诱导嵌合体重塑致癌激酶以触发细胞凋亡

Merz Manuel L, Shoba Veronika M, Pergu Rajaiah, Severance Zachary C, Munkanatta Godage Dhanushka N P, Deb Arghya, Kwok Hui Si, Singh Prashant, Singh Sameek, Allen Jonathan B, Tian Wenzhi, Gosavi Pallavi M, Chaudhary Santosh K, Anokhina Viktoriya, Weisberg Ellen L, Payne N Connor, He Yao, Osadchey Reilly, Shekhar Mrinal, Mazitschek Ralph, Rees Matthew G, Roth Jennifer A, Cui Qiang, Griffin James D, Liau Brian B, Choudhary Amit

Asymmetric Engagement of Dimeric CRL3 (KBTBD4) by the Molecular Glue UM171 Licenses Degradation of HDAC1/2 Complexes

分子胶UM171与二聚体CRL3(KBTBD4)的不对称结合促进HDAC1/2复合物的降解

Yeo, Megan Jr; Zhang, Olivia; Xie, Xiaowen; Nam, Eunju; Payne, Neil Connor; Gosavi, Pallavi M; Kwok, Hui Si; Iram, Irtiza; Lee, Ceejay; Li, Jiaming; Chen, Nicholas J; Jiang, Hanjie; Wang, Zhipeng A; Lee, Kwangwoon; Mao, Haibin; Harry, Stefan A; Barakat, Idris A; Takahashi, Mariko; Waterbury, Amanda L; Barone, Marco; Mattevi, Andrea; Bar-Peled, Liron; Cole, Philip A; Mazitschek, Ralph; Liau, Brian B; Zheng, Ning

Profiling the Landscape of Drug Resistance Mutations in Neosubstrates to Molecular Glue Degraders

分析新底物到分子胶降解剂的耐药突变图谱

Gosavi, Pallavi M; Ngan, Kevin C; Yeo, Megan J R; Su, Cindy; Li, Jiaming; Lue, Nicholas Z; Hoenig, Samuel M; Liau, Brian B

A Designed Enzyme Promotes Selective Post-translational Acylation

一种设计的酶促进选择性翻译后酰化

Gosavi, Pallavi M; Jayachandran, Megha; Rempillo, Joel J L; Zozulia, Oleksii; Makhlynets, Olga V; Korendovych, Ivan V

Short Self-Assembling Peptides Are Able to Bind to Copper and Activate Oxygen

短链自组装肽能够与铜结合并激活氧

Makhlynets, Olga V; Gosavi, Pallavi M; Korendovych, Ivan V

Functional characterization of a melittin analog containing a non-natural tryptophan analog

对含有非天然色氨酸类似物的蜂毒肽类似物进行功能表征

Ridgway, Zachary; Picciano, Angela L; Gosavi, Pallavi M; Moroz, Yurii S; Angevine, Christopher E; Chavis, Amy E; Reiner, Joseph E; Korendovych, Ivan V; Caputo, Gregory A