日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Conformational diversity in class C GPCR positive allosteric modulation.

C类GPCR正变构调节的构象多样性

Cannone Giuseppe, Berto Ludovic, Malhaire Fanny, Ferguson Gavin, Fouillen Aurelien, Balor Stéphanie, Font-Ingles Joan, Llebaria Amadeu, Goudet Cyril, Kotecha Abhay, K R Vinothkumar, Lebon Guillaume

Turn up the Vitamin D ReceptorNot the Calcium! Photoswitchable Vitamin D Agonists for Psoriasis

提高维生素D受体水平——而不是钙水平!用于治疗银屑病的维生素D光敏激动剂

Goudet, Cyril; Vázquez, Olalla

Mechanistic Insights into Light-Driven Allosteric Control of GPCR Biological Activity

光驱动变构调控GPCR生物活性的机制研究

Ricart-Ortega, Maria; Berizzi, Alice E; Pereira, Vanessa; Malhaire, Fanny; Catena, Juanlo; Font, Joan; Gómez-Santacana, Xavier; Muñoz, Lourdes; Zussy, Charleine; Serra, Carmen; Rovira, Xavier; Goudet, Cyril; Llebaria, Amadeu

Correction: Optical control of pain in vivo with a photoactive mGlu5 receptor negative allosteric modulator

更正:利用光敏mGlu5受体负变构调节剂对体内疼痛进行光学控制

Font, Joan; López-Cano, Marc; Notartomaso, Serena; Scarselli, Pamela; Di Prieto, Paola; Bresolí-Obach, Roger; Battaglia, Giuseppe; Malhaire, Fanny; Rovira, Xavier; Catena, Juanlo; Giraldo, Jesús; Pin, Jean-Philippe; Fernández-Dueñas, Víctor; Goudet, Cyril; Nonell, Santi; Nicoletti, Ferdinando; Llebaria, Amadeu; Ciruela, Francisco

Illuminating Phenylazopyridines To Photoswitch Metabotropic Glutamate Receptors: From the Flask to the Animals

利用光敏苯基偶氮吡啶类化合物调控代谢型谷氨酸受体:从烧瓶到动物实验

Gómez-Santacana, Xavier; Pittolo, Silvia; Rovira, Xavier; Lopez, Marc; Zussy, Charleine; Dalton, James A R; Faucherre, Adèle; Jopling, Chris; Pin, Jean-Philippe; Ciruela, Francisco; Goudet, Cyril; Giraldo, Jesús; Gorostiza, Pau; Llebaria, Amadeu

Allosteric control of an asymmetric transduction in a G protein-coupled receptor heterodimer.

G蛋白偶联受体异二聚体中不对称转导的变构控制

Liu Junke, Zhang Zongyong, Moreno-Delgado David, Dalton James Ar, Rovira Xavier, Trapero Ana, Goudet Cyril, Llebaria Amadeu, Giraldo Jesús, Yuan Qilin, Rondard Philippe, Huang Siluo, Liu Jianfeng, Pin Jean-Philippe

Shining Light on an mGlu5 Photoswitchable NAM: A Theoretical Perspective

揭示mGlu5光开关NAM的奥秘:理论视角

Dalton, James A R; Lans, Isaias; Rovira, Xavier; Malhaire, Fanny; Gómez-Santacana, Xavier; Pittolo, Silvia; Gorostiza, Pau; Llebaria, Amadeu; Goudet, Cyril; Pin, Jean-Philippe; Giraldo, Jesús

Evidence for a single heptahelical domain being turned on upon activation of a dimeric GPCR

证据表明,二聚体GPCR激活后,单个七螺旋结构域会被激活。

Hlavackova, Veronika; Goudet, Cyril; Kniazeff, Julie; Zikova, Alice; Maurel, Damien; Vol, Claire; Trojanova, Johana; Prézeau, Laurent; Pin, Jean-Philippe; Blahos, Jaroslav

Asymmetric functioning of dimeric metabotropic glutamate receptors disclosed by positive allosteric modulators

正向变构调节剂揭示二聚体代谢型谷氨酸受体的不对称功能

Goudet, Cyril; Kniazeff, Julie; Hlavackova, Veronika; Malhaire, Fanny; Maurel, Damien; Acher, Francine; Blahos, Jaroslav; Prézeau, Laurent; Pin, Jean-Philippe