日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Synthesis and Structure-Activity Relationship of Covalent Inhibitors of SARS-CoV-2 Papain-Like Protease with Antiviral Potency

SARS-CoV-2木瓜蛋白酶样蛋白酶共价抑制剂的合成及构效关系及其抗病毒活性

Rouch, Catherine C; Chatterjee, Arnab K; McCarty, Connor; Song, Lirui; Chu, Alan; Johnson, Kristen; Heacock, Mina; Riva, Laura; McNamara, Case W; Wolff, Karen C; Greene-Cramer, Rebecca; Falco, Anna De; Montelione, Gaetano T; Grabovyi, Gennadii A

Scalable Thiol Reactivity Profiling Identifies Azetidinyl Oxadiazoles as Cysteine-Targeting Electrophiles

可扩展的硫醇反应性分析表明,氮杂环丁基噁二唑是半胱氨酸靶向亲电试剂。

Ghorbani, Fereshte; You, Shaochen; Grabovyi, Gennadii A; Hong, Mannkyu; Lindsey, Garrett; Chatterjee, Arnab K; Bollong, Michael J

Discovery of CMX990: A Potent SARS-CoV-2 3CL Protease Inhibitor Bearing a Novel Warhead

CMX990 的发现:一种带有新型弹头的强效 SARS-CoV-2 3CL 蛋白酶抑制剂

Dayan Elshan, N G R; Wolff, Karen C; Riva, Laura; Woods, Ashley K; Grabovyi, Gennadii; Wilson, Katy; Pedroarena, James; Ghorai, Sourav; Nazarian, Armen; Weiss, Frank; Liu, Yuyin; Mazumdar, Wrickban; Song, Lirui; Okwor, Neechi; Malvin, Jacqueline; Bakowski, Malina A; Beutler, Nathan; Kirkpatrick, Melanie G; Gebara-Lamb, Amal; Huang, Edward; Nguyen-Tran, Vân T B; Chi, Victor; Li, Shuangwei; Rogers, Thomas F; McNamara, Case W; Gupta, Anil Kumar; Rahimi, Alireza; Chen, Jian Jeffrey; Joseph, Sean B; Schultz, Peter G; Chatterjee, Arnab K

Correction to "Discovery of CMX990: A Potent SARS-CoV-2 3CL Protease Inhibitor Bearing a Novel Warhead"

对“CMX990的发现:一种带有新型弹头的强效SARS-CoV-2 3CL蛋白酶抑制剂”一文的更正

Elshan, N G R Dayan; Wolff, Karen C; Riva, Laura; Woods, Ashley K; Grabovyi, Gennadii; Wilson, Katy; Pedroarena, James; Ghorai, Sourav; Nazarian, Armen; Weiss, Frank; Liu, Yuyin; Mazumdar, Wrickban; Song, Lirui; Okwor, Neechi; Malvin, Jacqueline; Liu, Dongdong; Bakowski, Malina A; Beutler, Nathan; Kirkpatrick, Melanie G; Gebara-Lamb, Amal; Huang, Edward; Nguyen-Tran, Vân T B; Chi, Victor; Li, Shuangwei; Rogers, Thomas F; McNamara, Case W; Gupta, Anil Kumar; Rahimi, Alireza; Chen, Jian Jeffrey; Joseph, Sean B; Schultz, Peter G; Chatterjee, Arnab K

Short Enantioselective Formal Synthesis of (-)-Platencin

(-)-Platencin 的简短对映选择性形式合成

Christian Defieber, Justin T Mohr, Gennadii A Grabovyi, Brian M Stoltz