Aminopyrazole Carboxamide Bruton's Tyrosine Kinase Inhibitors. Irreversible to Reversible Covalent Reactive Group Tuning
氨基吡唑羧酰胺类布鲁顿酪氨酸激酶抑制剂。不可逆到可逆共价反应基团调控
期刊:ACS Medicinal Chemistry Letters
影响因子:4
doi:10.1021/acsmedchemlett.8b00461
Schnute, Mark E; Benoit, Stephen E; Buchler, Ingrid P; Caspers, Nicole; Grapperhaus, Margaret L; Han, Seungil; Hotchandani, Rajeev; Huang, Nelson; Hughes, Robert O; Juba, Brian M; Kim, Kyung-Hee; Liu, Erica; McCarthy, Erin; Messing, Dean; Miyashiro, Joy S; Mohan, Shashi; O'Connell, Thomas N; Ohren, Jeffrey F; Parikh, Mihir D; Schmidt, Michelle; Selness, Shaun R; Springer, John R; Thanabal, Venkataraman; Trujillo, John I; Walker, Daniel P; Wan, Zhao-Kui; Withka, Jane M; Wittwer, Arthur J; Wood, Nancy L; Xing, Li; Zapf, Christoph W; Douhan, John 3rd