Leveraging Kinase Drugs for Neurosciences: Discovery of Selective, CNS-Penetrant Reversible Bruton's Tyrosine Kinase Inhibitors as Therapeutics for Neuroinflammation
利用激酶药物治疗神经科学:发现选择性、可穿透血脑屏障的可逆性布鲁顿酪氨酸激酶抑制剂作为神经炎症的治疗药物
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.5c02648
Hopkins, Brian T; Marx, Isaac E; Vandeveer, Harlod George; Nevalainen, Marta; Basile, Rebecca; Bajrami, Bekim; Choi, Colin K; Grater, Richard J; Gu, Chungang; Hoemberger, Marc; Kadakia, Ekta; Kapadnis, Sudarshan K; Liu, Ying; Ma, Bin; Magee, Tom; Metrick, Claire M; Mingueneau, Michael; Muste, Cathy A; Parker Harp, Chelsea R; Prince, Robin J; Santoro, Joseph C; Schulz, Jurgen; Sciabola, Simone; Tang, Hao; Wang, Ti; Meissner, Robert; Bohnert, Tonika
信号转导
炎症/感染
神经科学
神经炎症
血脑屏障
Neuroscience
炎症