Discovery of Tetrahydropyrazolopyridine as Sphingosine 1-Phosphate Receptor 3 (S1P3)-Sparing S1P1 Agonists Active at Low Oral Doses
发现四氢吡唑并吡啶作为鞘氨醇 1-磷酸受体 3 (S1P3) - 抑制 S1P1 激动剂,低口服剂量即可发挥作用
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.5b01512
Emmanuel H Demont, James M Bailey, Rino A Bit, Jack A Brown, Colin A Campbell, Nigel Deeks, Simon J Dowell, Colin Eldred, Pam Gaskin, James R J Gray, Andrea Haynes, David J Hirst, Duncan S Holmes, Umesh Kumar, Mary A Morse, Greg J Osborne, Jessica F Renaux, Gail A L Seal, Chris A Smethurst, Simon Ta