日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of Palazestrant (OP-1250), a Potent and Orally Bioavailable Complete Estrogen Receptor Antagonist (CERAN) and Selective Estrogen Receptor Degrader (SERD).

发现帕拉塞斯特兰(OP-1250),一种强效且口服生物利用度高的完全雌激素受体拮抗剂(CERAN)和选择性雌激素受体降解剂(SERD)

Ng Raymond A, Barratt Susanna, Parisian Alison, Palanisamy Gopinath S, Phukan Samiron, Sun Richard, Robello Brandon, Peña Guadalupe, Sapugay Judevin, Yeghikyan David, Wang Chenbo, Satish Kher Samir, Thangathirupathy Srinivasan, Millikin Robert, Yu Guijun, Watanabe Teruki, Zhou Fei, Rich Brian, Duncan Alexis, Andersen Samuel E, Chawla Reena, Zak David R, Heerding Dirk A, Hearn Brian R, Greene Geoffrey, Harmon Cyrus L, Hodges-Gallagher Leslie, Kushner Peter J, Fanning Sean W, Myles David C

Progesterone receptors drive advanced breast cancer phenotypes including circulating tumor- and stem-like cell expansion in the context of ESR1 mutation

在ESR1突变的情况下,孕激素受体驱动晚期乳腺癌表型,包括循环肿瘤细胞和干细胞样细胞的扩增。

Truong, Thu H; Gillis, Noelle E; Dwyer, Amy R; Huggins, Rosemary J; Hagen, Kyla M; Posani, Sai Harshita; Temiz, Nuri A; Kerkvliet, Carlos Perez; Piepgras, Ellie M; Ostrander, Julie H; Greene, Geoffrey L; Lange, Carol A

Ceramide-induced Endoplasmic Reticulum Stress as a Targetable Vulnerability in Endocrine Therapy-Resistant Breast Cancer.

神经酰胺诱导的内质网应激是内分泌治疗耐药性乳腺癌的一个可靶向脆弱性

Pal Purab, Chitkara Shweta, Sarpey Godwin K, Alani Fatimah, Zhao Huiping, Ata Malik, Qu Jun, Schiff Rachel, Tonetti Debra, Greene Geoffrey L, Frasor Jonna, Atilla-Gokcumen Gunes Ekin, Coloff Jonathan L

The relationship between fat distribution and diabetes in US adults by race/ethnicity

美国成年人脂肪分布与糖尿病的关系(按种族/族裔划分)

Xu, Furong; Earp, Jacob E; Riebe, Deborah; Delmonico, Matthew J; Lofgren, Ingrid E; Greene, Geoffrey W

FRI458 Rare Pathogenic Missense Variants in LMNA Identified in Women with Polycystic Ovary Syndrome (PCOS)

在多囊卵巢综合征(PCOS)女性中发现LMNA基因的FRI458罕见致病性错义变异

Paknikar, Raghavendra; Alpert, Lindsay; Cohen, Russell D; Shogan, Benjamin; Micic, Dejan; Muralidharan, Charanya; Huiping huang, Fei; May, Sarah C; Enriquez, Jacob; Nelson, Jennifer B; Wang, Eugenia; Chakraborthy, Advaita; Figatner, Kayla T; Navitskaya, Svetlana N; Tersey, Sarah A; Mirmira, Raghavendra G; Naaman, Sandra; Sintetas, Stephanie; Van Cauter, Eve; Hanlon, Erin C; Chopra, Karishma A; Gunaratne, Naiomi C; Deplewski, Dianne; Vallet, Amandine; Diennet, Marine; Thiombane, Khady; Vivet, Anaïs; Weber, Sandra; El Ezzy, Mohamed; Shaikh, Faraz; Poupart, Julien; Mendoza-Sanchez, Rodrigo; Alexandra Schuetz, Doris; Marinier, Anne; Greene, Geoffrey L; William Fanning, Sean; Nathalie Mader, Sylvie; Rashied, Ammar; Cursio, John; Hanlon, Erin C; Pannain, Silvana; Cipriani, Nicole A; Antic, Tatjana; Banizs, Anna; Finkelstein, Sydney David; Darji, Monika; Pannain, Silvana; Sam, Susan; Van Cauter, Eve; Hanlon, Erin C; Checkcinco, Christian; Tersey, Sarah A; Mirmira, Raghavendra G; Auckley, Elizabeth Diane; Arosemena, Marilyn A; Philipson, Louis; Ettleson, Matthew D; Laiteerapong, Neda; Wan, Wen; Bianco, Antonio C; Vasavada, Sheel R; Chopra, Karishma A; Philipson, Louis; Reutrakul, Sirimon; McAnany, J Jason; Park, Jason C; Chau, Felix Y; Danielson, Kirstie K; Bharati, Prasad; Pannain, Silvana; Van Cauter, Eve; Hanlon, Erin C; Freeman, Stephen J; Radonski, Brandon; Lecka, Liam; Davis, Ka'Derricka; Prince, Grace; Carthy, Kevin; Seley, Jane J; Song, Jing; Lee, Jungwha; Bailey, Stacy C; Khorzad, Rebeca; Gatchell, David; Ankenman, Bruce; Lewis, Daniel R; Holl, Jane; Wallia, Amisha; Salas Lucia, Federico; Hui Liao, Xiao; Jiang, Hanzi; Dumitrescu, Alexandra M; Refetoff, Samuel; Anselmo, Joao; Myong, Subin; Challa, Sridevi; Desai, Jui; Letourneau-Freiberg, Lisa; Msall, Michael; Scott, Megan; Nicole Naylor, Rochelle; Philipson, Louis; Greeley, Siri Atma W; Anderson, Cara; Kulkarni, Abhishek; Maier, Bernhard; Tersey, Sarah A; Anderson, Ryan; Mirmira, Raghavendra G; Ermis, Ebru; Nargis, Titli; Kulkarni, Abhishek; May, Sarah; Tersey, Sarah A; Mirmira, Raghavendra G; Anderson, Ryan M; Webster, Kierstin L; Wu, Wenting; Webb-Robertson, Bobbie-Jo; Nakayasu, Ernesto; Sarkar, Soumyadeep; Evans-Molina, Carmella; Tersey, Sarah A; Enriquez, Jacob; Hammes, Stephen R; Mirmira, Raghavendra G; Yang, Qiwei; Al-Hendy, Ayman; Bullock, Cydney A; Davis, Ka'Derricka; Carthy, Kevin; Wax, Pamela; Smyrniotis, Colleen; Pollack, Teresa; Barnard, Cynthia; Holl, Jane; Wallia, Amisha; Hammoud, Batoul; DiMeglio, Linda A; Kulkarni, Abishek; Hull, Audrey; Woerner, Stephanie; Cabrera, Susanne; Mastrandrea, Lucy D; Ouyang, Fangian; Perkins, Susan N; Evans-Molina, Carmella; Mastracci, Teresa L; Tersey, Sarah A; Sarkar, Soumyaddep; Nakayasu, Ernesto; Webb-Robertson, Bobbie-Jo; Gerner, Eugene; Mirmira, Raghavendra G; Sims, Emily K; Clarke, Bart; Aziz Khan, Aliya; Ruth Rubin, Mishaela; Schwarz, Peter E; Vokes, Tamara J; Shoback, Dolores M; Gagnon, Claudia; Palermo, Andrea; Abbott, Lisa G; Hofbauer, Lorenz C; Kohlmeier, Lynn; Cetani, Filomena; Phil, Susanne; An, Xuebei; Raymond Smith, Alden; Lai, Bryant; Le, John; Ukena, Jenny; Sibley, Christopher; Shu, Aimee; Rejnmark, Lars; Hancock, Govinda; Young, Kristen; Greene, Geoffrey L; Fanning, Sean William; Arosemena, Marilyn A; Wroblewski, Kristen; Tasali, Esra; Philipson, Louis H; Baboun, Daniela; Solano, Natalia; Sanchez, Andrea Martinez; Brathwaite, Carole; Restrepo, Ricardo; Alkhoury, Fuad; Carrillo-Iregui, Adriana; Li, Yanliang; Danielson, Kirstie K; Changhum Park, Jason; McAnany, J Jason; Chau, Felix Y; Prasad, Bharati; Hanlon, Erin C; Reutrakul, Sirimon; Salas Lucia, Federico; Dumitrescu, Alexandra M; Refetoff, Samuel; huang, fei; Nelson, Jennifer; Muralidharan, Charanya; Nakayasu, Ernesto; Yi, Xiaoyan; Eizirik, Decio; May, Sarah; Tersey, Sarah A; Mirmira, Raghavendra G; Nargis, Titli; Chakraborty, Advaita; Figatner, Kayla; Maloney, David; Boxer, Matthew; Tersey, Sarah A; Mirmira, Raghavendra G; Sidhu, Gurmanpreet; Madahar, Inderpreet; Haider, Adnan; Giordano, Jennifer; Liu, Jannel; Angelos, Peter; Barhoum, Maan; Jain, Rajesh; Kim, Keun Young; Hwang, Jessica; Sam, Susan; Bauer, Rosemary; Gorsic, Lidija; Legro, Richard S; Ehrmann, David; Geoffrey Hayes, M; Urbanek, Margrit

Dynamic epi-transcriptomic landscape mapping with disease progression in estrogen receptor-positive breast cancer

雌激素受体阳性乳腺癌疾病进展的动态表观转录组图谱绘制

Keelan, Stephen; Ola, Mihaela; Charmsaz, Sara; Cocchiglia, Sinéad; Ottaviani, Daniela; Hickey, Seán; Purcell, Siobhan; Bane, Fiona; Hegarty, Aisling; Doherty, Ben; Sheehan, Katherine; Hudson, Lance; Cosgrove, Nicola; Roux, Benjamin; Laine, Muriel; Greene, Geoffrey; Varešlija, Damir; Hill, Arnold Konrad; Young, Leonie

Reinvestigating the Synthesis and Characterization of Ethyl 3-[5-(2-Ethoxycarbonyl-1-methylvinyloxy)-1-methyl-1H-indol-3-yl]-but-2-enoate

重新研究3-[5-(2-乙氧羰基-1-甲基乙烯氧基)-1-甲基-1H-吲哚-3-基]-丁-2-烯酸乙酯的合成和表征

Li, Nan-Sheng; Piccirilli, Joseph A; Greene, Geoffrey L

Demethylation of dimethyl phosphonate esters with sodium ethanethiolate: Improved synthesis of 5'-methylene substituted 2',5'-deoxyribonucleotides

用乙硫醇钠对二甲基膦酸酯进行脱甲基化:改进的5'-亚甲基取代的2',5'-脱氧核苷酸的合成

Li, Nan-Sheng; Piccirilli, Joseph A; Greene, Geoffrey L

Stereospecific lasofoxifene derivatives reveal the interplay between estrogen receptor alpha stability and antagonistic activity in ESR1 mutant breast cancer cells

立体特异性拉索昔芬衍生物揭示了雌激素受体α稳定性与ESR1突变型乳腺癌细胞拮抗活性之间的相互作用

Hosfield, David J; Weber, Sandra; Li, Nan-Sheng; Sauvage, Madline; Joiner, Carstyn F; Hancock, Govinda R; Sullivan, Emily A; Ndukwe, Estelle; Han, Ross; Cush, Sydney; Lainé, Muriel; Mader, Sylvie C; Greene, Geoffrey L; Fanning, Sean W

The Relationship of Physical Activity and Dietary Quality with Android Fat Composition and Distribution in US Adults

美国成年人体力活动和饮食质量与安卓脂肪组成和分布的关系

Xu, Furong; Earp, Jacob E; LoBuono, Dara L; Greene, Geoffrey W