日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Hydroxamate-based inhibitors reveal structural determinants of selectivity for Plasmodium falciparum aminopeptidase P

基于羟肟酸酯的抑制剂揭示了恶性疟原虫氨肽酶P选择性的结构决定因素

Mills, Belinda J; Gregory, Kyle S; Cozier, Gyles E; Taweechai, Supannee; Loughlan, Eve; McConkey, Glenn A; Isaac, R Elwyn; Foster, Richard; Acharya, K Ravi

Molecular basis of domain-specific angiotensin I-converting enzyme inhibition by the antihypertensive drugs enalaprilat, ramiprilat, trandolaprilat, quinaprilat and perindoprilat

抗高血压药物依那普利拉、雷米普利拉、群多普利拉、喹那普利拉和培哚普利拉对血管紧张素I转化酶的结构域特异性抑制的分子基础

Gregory, Kyle S; Ramasamy, Vinasha; Sturrock, Edward D; Acharya, K Ravi

Molecular Basis of Dipeptide Recognition in Drosophila melanogaster Angiotensin I-Converting Enzyme Homologue, AnCE

果蝇血管紧张素I转化酶同源物(AnCE)中二肽识别的分子基础

Żukowska, Joanna; Gregory, Kyle S; Robinson, Adam; Isaac, R Elwyn; Acharya, K Ravi

Ciprofloxacin Inhibits Angiotensin I‑Converting Enzyme (ACE) Activity by Binding at the Exosite, Distal to the Catalytic Pocket

环丙沙星通过与催化口袋远端的外位点结合来抑制血管紧张素I转化酶(ACE)的活性。

Gregory, Kyle S; Ramasamy, Vinasha; Sturrock, Edward D; Acharya, K Ravi

Molecular basis of human angiotensin-1 converting enzyme inhibition by a series of diprolyl-derived compounds

二丙二酰基衍生物抑制人血管紧张素-1转化酶的分子机制

Gregory, Kyle S; Cozier, Gyles E; Fienberg, Stephen; Chibale, Kelly; Sturrock, Edward D; Acharya, K Ravi

Advances in the structural basis for angiotensin-1 converting enzyme (ACE) inhibitors

血管紧张素-1转化酶(ACE)抑制剂结构基础的研究进展

Acharya, K Ravi; Gregory, Kyle S; Sturrock, Edward D

Crystal Structure of the Catalytic Domain of a Botulinum Neurotoxin Homologue from Enterococcus faecium: Potential Insights into Substrate Recognition

粪肠球菌肉毒杆菌神经毒素同源物催化结构域的晶体结构:对底物识别的潜在启示

Gregory, Kyle S; Hall, Peter-Rory; Onuh, Jude Prince; Mojanaga, Otsile O; Liu, Sai Man; Acharya, K Ravi

A Molecular Analysis of the Aminopeptidase P-Related Domain of PID-5 from Caenorhabditis elegans

秀丽隐杆线虫PID-5氨肽酶P相关结构域的分子分析

Lloyd, Anna C; Gregory, Kyle S; Isaac, R Elwyn; Acharya, K Ravi

A Comprehensive Structural Analysis of Clostridium botulinum Neurotoxin A Cell-Binding Domain from Different Subtypes

不同亚型肉毒梭菌神经毒素A细胞结合域的综合结构分析

Gregory, Kyle S; Acharya, K Ravi

Crystal Structures of Botulinum Neurotoxin Subtypes A4 and A5 Cell Binding Domains in Complex with Receptor Ganglioside

肉毒杆菌神经毒素A4和A5亚型细胞结合域与受体神经节苷脂复合物的晶体结构

Gregory, Kyle S; Mojanaga, Otsile O; Liu, Sai Man; Acharya, K Ravi