Pseudo-cyclization through intramolecular hydrogen bond enables discovery of pyridine substituted pyrimidines as new Mer kinase inhibitors
通过分子内氢键进行伪环化,发现吡啶取代的嘧啶作为新的 Mer 激酶抑制剂
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/jm401387j
Weihe Zhang, Dehui Zhang, Michael A Stashko, Deborah DeRyckere, Debra Hunter, Dmitri Kireev, Michael J Miley, Christopher Cummings, Minjung Lee, Jacqueline Norris-Drouin, Wendy M Stewart, Susan Sather, Yingqiu Zhou, Gregory Kirkpatrick, Mischa Machius, William P Janzen, H Shelton Earp, Douglas K Gra